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Refinado por: Nome da Publicação: Bioorganic & Medicinal Chemistry Letters remover
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1
Synthesis and biological evaluation of DIDS analogues as efficient inhibitors of RAD51 involved in homologous recombination
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Artigo
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Synthesis and biological evaluation of DIDS analogues as efficient inhibitors of RAD51 involved in homologous recombination

Demeyer, Alexandre ; Fonteneau, Lucie ; Liennard, Marion ; Foyer, Claire ; Weigel, Pierre ; Laurent, Adèle D. ; Lebreton, Jacques ; Fleury, Fabrice ; Mathé-Allainmat, Monique

Bioorganic & medicinal chemistry letters, 2023-05, Vol.87, p.129261-129261, Article 129261 [Periódico revisado por pares]

England: Elsevier Ltd

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2
Substitution of a triazole for the central olefin in biologically active stilbenes
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Artigo
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Substitution of a triazole for the central olefin in biologically active stilbenes

Stockdale, David P. ; Beutler, John A. ; Wiemer, David F.

Bioorganic & medicinal chemistry letters, 2022-11, Vol.75, p.128980-128980, Article 128980 [Periódico revisado por pares]

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3
Synthesis and biological evaluation of substituted amide derivatives of C4-ageratochromene dimer analog
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Artigo
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Synthesis and biological evaluation of substituted amide derivatives of C4-ageratochromene dimer analog

Agarwal, Karishma ; Gupta, Kratika ; Sharma, Kriti ; Khanka, Sonu ; Singh, Shilpi ; Singh, Jyoti ; Trivedi, Laxmikant ; Vasdev, Prema G. ; Luqman, Suaib ; Khan, Feroz ; Singh, Divya ; Gupta, Atul

Bioorganic & medicinal chemistry letters, 2021-10, Vol.50, p.128340-128340, Article 128340 [Periódico revisado por pares]

England: Elsevier Ltd

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4
Mur ligases inhibitors with azastilbene scaffold: Expanding the structure–activity relationship
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Artigo
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Mur ligases inhibitors with azastilbene scaffold: Expanding the structure–activity relationship

Hrast, Martina ; Frlan, Rok ; Knez, Damijan ; Zdovc, Irena ; Barreteau, Hélène ; Gobec, Stanislav

Bioorganic & medicinal chemistry letters, 2021-05, Vol.40, p.127966-127966, Article 127966 [Periódico revisado por pares]

England: Elsevier Ltd

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5
Fluorescence properties of retinoid X receptor antagonist NEt-SB
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Artigo
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Fluorescence properties of retinoid X receptor antagonist NEt-SB

Yamada, Shoya ; Takamura, Yuta ; Fujihara, Michiko ; Kawasaki, Mayu ; Ito, Sohei ; Nakano, Shogo ; Kakuta, Hiroki

Bioorganic & medicinal chemistry letters, 2021-01, Vol.31, p.127666-127666, Article 127666 [Periódico revisado por pares]

England: Elsevier Ltd

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6
Induced osteoblast differentiation by amide derivatives of stilbene: The possible osteogenic agents
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Artigo
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Induced osteoblast differentiation by amide derivatives of stilbene: The possible osteogenic agents

Imran Ahamad, Mohd ; Prakash, Ravi ; John, Aijaz A ; Wani, Zahoor ; Yadav, Deepika ; Bawankule, Dnyaneshwar U. ; Luqman, Suaib ; Khan, Feroz ; Singh, Divya ; Gupta, Atul

Bioorganic & medicinal chemistry letters, 2020-06, Vol.30 (11), p.127138-127138, Article 127138 [Periódico revisado por pares]

England: Elsevier Ltd

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7
Tetra-aryl cyclobutane and stilbenes from the rhizomes of Rheum undulatum and their α-glucosidase inhibitory activity: Biological evaluation, kinetic analysis, and molecular docking simulation
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Artigo
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Tetra-aryl cyclobutane and stilbenes from the rhizomes of Rheum undulatum and their α-glucosidase inhibitory activity: Biological evaluation, kinetic analysis, and molecular docking simulation

Ha, Manh Tuan ; Kim, Minji ; Kim, Chung Sub ; Park, Se-Eun ; Kim, Jeong Ah ; Woo, Mi Hee ; Choi, Jae Sue ; Min, Byung Sun

Bioorganic & medicinal chemistry letters, 2020-04, Vol.30 (8), p.127049, Article 127049 [Periódico revisado por pares]

England: Elsevier Ltd

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8
Synthesis and biological evaluation of novel pyrazolo[3,4-b]pyridines as cis-restricted combretastatin A-4 analogues
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Artigo
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Synthesis and biological evaluation of novel pyrazolo[3,4-b]pyridines as cis-restricted combretastatin A-4 analogues

Jian, Xie-Er ; Yang, Fang ; Jiang, Cui-Shan ; You, Wen-Wei ; Zhao, Pei-Liang

Bioorganic & medicinal chemistry letters, 2020-04, Vol.30 (8), p.127025, Article 127025 [Periódico revisado por pares]

England: Elsevier Ltd

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9
Design and synthesis of (E)-1,2-diphenylethene-based EZH2 inhibitors
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Artigo
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Design and synthesis of (E)-1,2-diphenylethene-based EZH2 inhibitors

He, Hualong ; Hu, Xi ; Teng, Fei ; Liu, Zhihao ; Zhang, Qiangsheng ; Feng, Zhanzhan ; Feng, Qiang ; Yu, Luoting

Bioorganic & medicinal chemistry letters, 2020-03, Vol.30 (5), p.126957, Article 126957 [Periódico revisado por pares]

England: Elsevier Ltd

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10
Comparative analysis of stilbene and benzofuran neolignan derivatives as acetylcholinesterase inhibitors with neuroprotective and anti-inflammatory activities
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Artigo
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Comparative analysis of stilbene and benzofuran neolignan derivatives as acetylcholinesterase inhibitors with neuroprotective and anti-inflammatory activities

Nagumo, Mina ; Ninomiya, Masayuki ; Oshima, Natsuko ; Itoh, Tomohiro ; Tanaka, Kaori ; Nishina, Atsuyoshi ; Koketsu, Mamoru

Bioorganic & medicinal chemistry letters, 2019-09, Vol.29 (17), p.2475-2479 [Periódico revisado por pares]

England: Elsevier Ltd

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