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Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies

Yeung, Kap-Sun ; Beno, Brett R ; Parcella, Kyle ; Bender, John A ; Grant-Young, Katherine A ; Nickel, Andrew ; Gunaga, Prashantha ; Anjanappa, Prakash ; Bora, Rajesh Onkardas ; Selvakumar, Kumaravel ; Rigat, Karen ; Wang, Ying-Kai ; Liu, Mengping ; Lemm, Julie ; Mosure, Kathy ; Sheriff, Steven ; Wan, Changhong ; Witmer, Mark ; Kish, Kevin ; Hanumegowda, Umesh ; Zhuo, Xiaoliang ; Shu, Yue-Zhong ; Parker, Dawn ; Haskell, Roy ; Ng, Alicia ; Gao, Qi ; Colston, Elizabeth ; Raybon, Joseph ; Grasela, Dennis M ; Santone, Kenneth ; Gao, Min ; Meanwell, Nicholas A ; Sinz, Michael ; Soars, Matthew G ; Knipe, Jay O ; Roberts, Susan B ; Kadow, John F

Journal of medicinal chemistry, 2017-05, Vol.60 (10), p.4369-4385 [Periódico revisado por pares]

United States: American Chemical Society

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