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1
A FRET-based assay for the discovery of West Nile Virus NS2B-NS3 protease inhibitors
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Artigo
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A FRET-based assay for the discovery of West Nile Virus NS2B-NS3 protease inhibitors

Adamek, Rebecca N ; Maniquis, Roxanne V ; Khakoo, Sabaha ; Bridges, Michael D ; Salzameda, Nicholas T

Bioorganic & Medicinal Chemistry Letters, 2013-09, Vol.23 (17), p.4848-4850

eScholarship, University of California

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2
Resistance mutations of NS3 and NS5b in treatment-naïve patients infected with hepatitis C virus in Santa Catarina and Rio Grande do Sul states, Brazil
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Artigo
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Resistance mutations of NS3 and NS5b in treatment-naïve patients infected with hepatitis C virus in Santa Catarina and Rio Grande do Sul states, Brazil

Andrade, Elisabete ; Rocha, Daniele ; Fontana-Maurell, Marcela ; Costa, Elaine ; Ribeiro, Marisa ; Godoy, Daniela Tupy de ; Ferreira, Antonio G P ; Tanuri, Amilcar ; Brindeiro, Rodrigo ; Alvarez, Patrícia

Genetics and molecular biology, 2020-01, Vol.43 (1), p.e20180237-e20180237 [Periódico revisado por pares]

Brazil: Sociedade Brasileira de Genetica

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3
The design of potent, non-peptidic inhibitors of hepatitis C protease
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Artigo
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The design of potent, non-peptidic inhibitors of hepatitis C protease

Andrews, David M. ; Chaignot, Helene M. ; Coomber, Barry A. ; Dowle, Mike D. ; Lucy Hind, S. ; Johnson, Martin R. ; Jones, Paul S. ; Mills, Gail ; Patikis, Angela ; Pateman, Tony J. ; Ed Robinson, J. ; Slater, Martin J. ; Trivedi, Naimisha

European journal of medicinal chemistry, 2003-04, Vol.38 (4), p.339-343 [Periódico revisado por pares]

Oxford: Elsevier Masson SAS

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4
Antiviral Activity and Resistance Analysis of NS3/4A Protease Inhibitor Grazoprevir and NS5A Inhibitor Elbasvir in Hepatitis C Virus GT4 Replicons
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Artigo
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Antiviral Activity and Resistance Analysis of NS3/4A Protease Inhibitor Grazoprevir and NS5A Inhibitor Elbasvir in Hepatitis C Virus GT4 Replicons

Asante-Appiah, Ernest ; Curry, Stephanie ; McMonagle, Patricia ; Ingravallo, Paul ; Chase, Robert ; Nickle, David ; Qiu, Ping ; Howe, Anita ; Lahser, Frederick C

Antimicrobial agents and chemotherapy, 2017-07, Vol.61 (7) [Periódico revisado por pares]

United States: American Society for Microbiology

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5
The Design and Synthesis of Potent Inhibitors of Hepatitis C Virus NS3–4A Proteinase
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The Design and Synthesis of Potent Inhibitors of Hepatitis C Virus NS3–4A Proteinase

Attwood, MR ; Bennett, JM ; Campbell, AD ; Canning, GGM ; Carr, MG ; Conway, E ; Dunsdon, RM ; Greening, JR ; Jones, PS ; Kay, PB ; Handa, BK ; Hurst, DN ; Jennings, NS ; Jordan, S ; Keech, E ; O'Brien, MA ; Overton, HA ; King-Underwood, J ; Raynham, TM ; Stenson, KP ; Wilkinson, CS ; Wilkinson, TCI ; Wilson, FX

Antiviral chemistry & chemotherapy, 1999-09, Vol.10 (5), p.259-273 [Periódico revisado por pares]

London, England: SAGE Publications

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6
Inhibitors of hepatitis C virus NS3/4A: α-Ketoamide based macrocyclic inhibitors
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Inhibitors of hepatitis C virus NS3/4A: α-Ketoamide based macrocyclic inhibitors

Avolio, Salvatore ; Robertson, Keith ; Hernando, Josè Ignacio Martin ; DiMuzio, Jillian ; Summa, Vincenzo

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2295-2298 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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7
The Dimeric Peptide (KKYRYHLKPF)2K Shows Broad-Spectrum Antiviral Activity by Inhibiting Different Steps of Chikungunya and Zika Virus Infection
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Artigo
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The Dimeric Peptide (KKYRYHLKPF)2K Shows Broad-Spectrum Antiviral Activity by Inhibiting Different Steps of Chikungunya and Zika Virus Infection

Ayusso, Gabriela Miranda ; Lima, Maria Letícia Duarte ; da Silva Sanches, Paulo Ricardo ; Santos, Igor Andrade ; Martins, Daniel Oliveira Silva ; da Conceição, Pâmela Jóyce Previdelli ; Carvalho, Tamara ; da Costa, Vivaldo Gomes ; Bittar, Cíntia ; Merits, Andres ; Santos-Filho, Norival Alves ; Cilli, Eduardo Maffud ; Jardim, Ana Carolina Gomes ; de Freitas Calmon, Marilia ; Rahal, Paula

Viruses, 2023-05, Vol.15 (5), p.1168 [Periódico revisado por pares]

Basel: MDPI AG

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8
Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs
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Artigo
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Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs

Bäck, Marcus ; Johansson, Per-Ola ; Wångsell, Fredrik ; Thorstensson, Fredrik ; Kvarnström, Ingemar ; Ayesa, Susana ; Wähling, Horst ; Pelcman, Mikael ; Jansson, Katarina ; Lindström, Stefan ; Wallberg, Hans ; Classon, Björn ; Rydergård, Christina ; Vrang, Lotta ; Hamelink, Elizabeth ; Hallberg, Anders ; Rosenquist, Åsa ; Samuelsson, Bertil

Bioorganic & medicinal chemistry, 2007-11, Vol.15 (22), p.7184-7202 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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9
Extent of HCV NS3 protease variability and resistance-associated mutations assessed by next generation sequencing in HCV monoinfected and HIV/HCV coinfected patients
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Artigo
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Extent of HCV NS3 protease variability and resistance-associated mutations assessed by next generation sequencing in HCV monoinfected and HIV/HCV coinfected patients

Bartolini, Barbara ; Giombini, Emanuela ; Zaccaro, Paola ; Selleri, Marina ; Rozera, Gabriella ; Abbate, Isabella ; Comandini, Ubaldo Visco ; Ippolito, Giuseppe ; Solmone, Mariacarmela ; Capobianchi, Maria R.

Virus research, 2013-11, Vol.177 (2), p.205-208 [Periódico revisado por pares]

Netherlands: Elsevier B.V

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10
Development of hepatitis C virus chimeric replicons for identifying broad spectrum NS3 protease inhibitors
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Development of hepatitis C virus chimeric replicons for identifying broad spectrum NS3 protease inhibitors

Binder, Joseph ; Tetangco, Selwyna ; Weinshank, Megan ; Maegley, Karen ; Lingardo, Laura ; Diehl, Wade ; Love, Robert ; Patick, Amy K. ; Smith, George J.

Antiviral research, 2011-08, Vol.91 (2), p.102-111 [Periódico revisado por pares]

Kidlington: Elsevier B.V

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