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1
In silico analysis and in vitro evaluation of immunogenic and immunomodulatory properties of promiscuous peptides derived from Leishmania infantum eukaryotic initiation factor
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In silico analysis and in vitro evaluation of immunogenic and immunomodulatory properties of promiscuous peptides derived from Leishmania infantum eukaryotic initiation factor

Koutsoni, Olga S. ; Routsias, John G. ; Kyriazis, Ioannis D. ; Barhoumi, Mourad ; Guizani, Ikram ; Tsakris, Athanassios ; Dotsika, Eleni

Bioorganic & medicinal chemistry, 2017-11, Vol.25 (21), p.5904-5916 [Periódico revisado por pares]

England: Elsevier Ltd

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2
N-Propargylpiperidines with naphthalene-2-carboxamide or naphthalene-2-sulfonamide moieties: Potential multifunctional anti-Alzheimer’s agents
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Artigo
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N-Propargylpiperidines with naphthalene-2-carboxamide or naphthalene-2-sulfonamide moieties: Potential multifunctional anti-Alzheimer’s agents

Košak, Urban ; Knez, Damijan ; Coquelle, Nicolas ; Brus, Boris ; Pišlar, Anja ; Nachon, Florian ; Brazzolotto, Xavier ; Kos, Janko ; Colletier, Jacques-Philippe ; Gobec, Stanislav

Bioorganic & medicinal chemistry, 2017-01, Vol.25 (2), p.633-645 [Periódico revisado por pares]

England: Elsevier Ltd

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3
Novel hydroxybenzylamine-deoxyvasicinone hybrids as anticholinesterase therapeutics for Alzheimer’s disease
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Artigo
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Novel hydroxybenzylamine-deoxyvasicinone hybrids as anticholinesterase therapeutics for Alzheimer’s disease

Bowroju, Suresh K. ; Penthala, Narsimha R. ; Lakkaniga, Naga Rajiv ; Balasubramaniam, Meenakshisundaram ; Ayyadevara, Srinivas ; Shmookler Reis, Robert J. ; Crooks, Peter A.

Bioorganic & medicinal chemistry, 2021-09, Vol.45, p.116311-116311, Article 116311 [Periódico revisado por pares]

England: Elsevier Ltd

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4
Self-assembly of photosensitive and radiotherapeutic peptide for combined photodynamic-radio cancer therapy with intracellular delivery of miRNA-139-5p
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Artigo
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Self-assembly of photosensitive and radiotherapeutic peptide for combined photodynamic-radio cancer therapy with intracellular delivery of miRNA-139-5p

Wang, Hanhua ; Wang, Ziyi ; Chen, Weiwei ; Wang, Wencai ; Shi, Woda ; Chen, Jinzhong ; Hang, Ye ; Song, Jin ; Xiao, Xiao ; Dai, Zhenyu

Bioorganic & medicinal chemistry, 2021-08, Vol.44, p.116305, Article 116305 [Periódico revisado por pares]

England: Elsevier Ltd

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5
Concise solid-phase synthesis enables derivatisation of YEATS domain cyclopeptide inhibitors for improved cellular uptake
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Artigo
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Concise solid-phase synthesis enables derivatisation of YEATS domain cyclopeptide inhibitors for improved cellular uptake

Jiang, Yixiang ; Liu, Sha ; Tian, Gaofei ; Cheung, Hayden Jit Hei ; Li, Xin ; Li, Xiang David

Bioorganic & medicinal chemistry, 2021-09, Vol.45, p.116342-116342, Article 116342 [Periódico revisado por pares]

England: Elsevier Ltd

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6
Lipidated α/Sulfono-α-AA heterogeneous peptides as antimicrobial agents for MRSA
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Artigo
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Lipidated α/Sulfono-α-AA heterogeneous peptides as antimicrobial agents for MRSA

Singh, Sylvia ; Wang, Minghui ; Gao, Ruixuan ; Teng, Peng ; Odom, Timothy ; Zhang, En ; Xu, Hai ; Cai, Jianfeng

Bioorganic & medicinal chemistry, 2020-01, Vol.28 (1), p.115241-115241, Article 115241 [Periódico revisado por pares]

England: Elsevier Ltd

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7
Small molecule mimics of DFTamP1, a database designed anti-Staphylococcal peptide
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Artigo
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Small molecule mimics of DFTamP1, a database designed anti-Staphylococcal peptide

Dong, Yuxiang ; Lushnikova, Tamara ; Golla, Radha M. ; Wang, Xiaofang ; Wang, Guangshun

Bioorganic & medicinal chemistry, 2017-02, Vol.25 (3), p.864-869 [Periódico revisado por pares]

England: Elsevier Ltd

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8
Biofunctional supramolecular hydrogels fabricated from a short self-assembling peptide modified with bioactive sequences for the 3D culture of breast cancer MCF-7 cells
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Biofunctional supramolecular hydrogels fabricated from a short self-assembling peptide modified with bioactive sequences for the 3D culture of breast cancer MCF-7 cells

Chia, Jyh Yea ; Miki, Takayuki ; Mihara, Hisakazu ; Tsutsumi, Hiroshi

Bioorganic & medicinal chemistry, 2021-09, Vol.46, p.116345-116345, Article 116345 [Periódico revisado por pares]

England: Elsevier Ltd

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9
Peptidomimetic analogues of an Arg-Trp-x-x-Trp motif responsible for interaction of translocase MraY with bacteriophage ϕX174 lysis protein E
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Artigo
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Peptidomimetic analogues of an Arg-Trp-x-x-Trp motif responsible for interaction of translocase MraY with bacteriophage ϕX174 lysis protein E

Kerr, Rachel V. ; Fairbairn, Julia A. ; Merritt, Andrew T. ; Bugg, Timothy D.H.

Bioorganic & medicinal chemistry, 2021-12, Vol.52, p.116502-116502, Article 116502 [Periódico revisado por pares]

England: Elsevier Ltd

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10
Stapled peptide-based membrane fusion inhibitors of hepatitis C virus
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Artigo
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Stapled peptide-based membrane fusion inhibitors of hepatitis C virus

Cui, Hong-Kui ; Qing, Jie ; Guo, Ye ; Wang, Yu-Jia ; Cui, Li-Jia ; He, Tian-Hua ; Zhang, Linqi ; Liu, Lei

Bioorganic & medicinal chemistry, 2013-06, Vol.21 (12), p.3547-3554 [Periódico revisado por pares]

England: Elsevier Ltd

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