Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor
Jean Francisco Rosa Ribeiro Lorenzo Cianni; Chan Li; Thomas G Warwick; Daniela de Vita; Fabiana Rosini; Fernanda dos Reis Rocho; Felipe Cardoso Prado Martins; Peter W Kenny; Jerônimo Lameira; Andrei Leitão; Jonas Emsley; Carlos Alberto Montanari
Bioorganic and Medicinal Chemistry Oxford : Elsevier v. 22, n. 22, p. 115743, November 2020
Oxford 2020
Localização:
IQSC - Inst. Química de São Carlos
(P19023 )(Acessar)
Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement
Juliana C Gomes Lorenzo Cianni; Jean Ribeiro; Fernanda dos Reis Rocho; Samelyn da Costa Martins Silva; Pedro Henrique J Batista; Carolina Borsoi Moraes; Caio Haddad Franco; Lúcio H G Freitas Junior; Peter W Kenny; Andrei Leitão; Antonio Carlos Bender Burtoloso; Daniela de Vita; Carlos Alberto Montanari
Bioorganic and Medicinal Chemistry Oxford: Elsevier Ltd v. 27, n. 22, p.x 115083, nov, 2019
Oxford 2019
Localização:
IQSC - Inst. Química de São Carlos
(P18260 )(Acessar)