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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists
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Artigo
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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists

Han, Sangdon ; Thoresen, Lars ; Zhu, Xiuwen ; Narayanan, Sanju ; Jung, Jae-Kyu ; Strah-Pleynet, Sonja ; Decaire, Marc ; Choi, Karoline ; Xiong, Yifeng ; Yue, Dawei ; Semple, Graeme ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Al-Shamma, Hussien ; Gatlin, Joel ; Chen, Ruoping ; Dang, Huong ; Pride, Cameron ; Gaidarov, Ibragim ; Unett, David J ; Behan, Dominic P ; Sadeque, Abu ; Usmani, Khawja A ; Chen, Chuan ; Edwards, Jeffrey ; Morgan, Michael ; Jones, Robert M

Bioorganic & medicinal chemistry letters, 2015-01, Vol.25 (2), p.322-326 [Periódico revisado por pares]

England

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2
Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxam i des as potent and selective CB sub(2) receptor agonists
Material Type:
Artigo
Adicionar ao Meu Espaço

Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxam i des as potent and selective CB sub(2) receptor agonists

Han, Sangdon ; Thoresen, Lars ; Zhu, Xiuwen ; Narayanan, Sanju ; Jung, Jae-Kyu ; Strah-Pleynet, Sonja ; Decaire, Marc ; Choi, Karoline ; Xiong, Yifeng ; Yue, Dawei ; Semple, Graeme ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Al-Shamma, Hussien ; Gatlin, Joel ; Chen, Ruoping ; Dang, Huong ; Pride, Cameron ; Gaidarov, Ibragim ; Unett, David J ; Behan, Dominic P ; Sadeque, Abu ; Usmani, Khawja A ; Chen, Chuan ; Edwards, Jeffrey ; Morgan, Michael ; Jones, Robert M

Bioorganic & medicinal chemistry letters, 2015-01, Vol.25 (2), p.322-326 [Periódico revisado por pares]

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3
Fused tricyclic indoles as S1P1 agonists with robust efficacy in animal models of autoimmune disease
Material Type:
Artigo
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Fused tricyclic indoles as S1P1 agonists with robust efficacy in animal models of autoimmune disease

Buzard, Daniel J. ; Han, Sangdon ; Lopez, Luis ; Kawasaki, Andrew ; Moody, Jeanne ; Thoresen, Lars ; Ullman, Brett ; Lehmann, Juerg ; Calderon, Imelda ; Zhu, Xiuwen ; Gharbaoui, Tawfik ; Sengupta, Dipanjan ; Krishnan, Ashwin ; Gao, Yinghong ; Edwards, Jeff ; Barden, Jeremy ; Morgan, Michael ; Usmani, Khawja ; Chen, Chuan ; Sadeque, Abu ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Liu, Ling ; Al-Shamma, Hussien ; Gatlin, Joel ; Le, Minh ; Xing, Charles ; Espinola, Sheryll ; Jones, Robert M.

Bioorganic & medicinal chemistry letters, 2012-07, Vol.22 (13), p.4404-4409 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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