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Refinado por: Nome da Publicação: Bioorganic & Medicinal Chemistry Letters remover autor: Whelan, Kevin remover autor: Fu, Lixia remover
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1
A new family of H3 receptor antagonists based on the natural product Conessine
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A new family of H3 receptor antagonists based on the natural product Conessine

SANTORA, Vincent J ; COVEL, Jonathan A ; WEBB, Robert R ; SAGE, Carleton ; REN, Albert ; PEREIRA, Guilherme ; KNUDSEN, Jens ; EDWARDS, Jeffrey E ; SUAREZ, Marissa ; FRAZER, John ; THOMSEN, William ; HAUSER, Erin ; HAYASHI, Rena ; WHELAN, Kevin ; GROTTICK, Andrew J ; HOFILENA, Brian J ; IBARRA, Jason B ; PULLEY, Michelle D ; WEINHOUSE, Michael I ; SENGUPTA, Dipanjan ; DUFFIELD, Jonathan J ; SEMPLE, Graeme

Bioorganic & medicinal chemistry letters, 2008-02, Vol.18 (4), p.1490-1494 [Periódico revisado por pares]

Oxford: Elsevier

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2
Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists
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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists

Han, Sangdon ; Thoresen, Lars ; Zhu, Xiuwen ; Narayanan, Sanju ; Jung, Jae-Kyu ; Strah-Pleynet, Sonja ; Decaire, Marc ; Choi, Karoline ; Xiong, Yifeng ; Yue, Dawei ; Semple, Graeme ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Al-Shamma, Hussien ; Gatlin, Joel ; Chen, Ruoping ; Dang, Huong ; Pride, Cameron ; Gaidarov, Ibragim ; Unett, David J ; Behan, Dominic P ; Sadeque, Abu ; Usmani, Khawja A ; Chen, Chuan ; Edwards, Jeffrey ; Morgan, Michael ; Jones, Robert M

Bioorganic & medicinal chemistry letters, 2015-01, Vol.25 (2), p.322-326 [Periódico revisado por pares]

England

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3
Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxam i des as potent and selective CB sub(2) receptor agonists
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Artigo
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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxam i des as potent and selective CB sub(2) receptor agonists

Han, Sangdon ; Thoresen, Lars ; Zhu, Xiuwen ; Narayanan, Sanju ; Jung, Jae-Kyu ; Strah-Pleynet, Sonja ; Decaire, Marc ; Choi, Karoline ; Xiong, Yifeng ; Yue, Dawei ; Semple, Graeme ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Al-Shamma, Hussien ; Gatlin, Joel ; Chen, Ruoping ; Dang, Huong ; Pride, Cameron ; Gaidarov, Ibragim ; Unett, David J ; Behan, Dominic P ; Sadeque, Abu ; Usmani, Khawja A ; Chen, Chuan ; Edwards, Jeffrey ; Morgan, Michael ; Jones, Robert M

Bioorganic & medicinal chemistry letters, 2015-01, Vol.25 (2), p.322-326 [Periódico revisado por pares]

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4
A new family of H 3 receptor antagonists based on the natural product Conessine
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Artigo
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A new family of H 3 receptor antagonists based on the natural product Conessine

Santora, Vincent J. ; Covel, Jonathan A. ; Hayashi, Rena ; Hofilena, Brian J. ; Ibarra, Jason B. ; Pulley, Michelle D. ; Weinhouse, Michael I. ; Sengupta, Dipanjan ; Duffield, Jonathan J. ; Semple, Graeme ; Webb, Robert R. ; Sage, Carleton ; Ren, Albert ; Pereira, Guilherme ; Knudsen, Jens ; Edwards, Jeffrey E. ; Suarez, Marissa ; Frazer, John ; Thomsen, William ; Hauser, Erin ; Whelan, Kevin ; Grottick, Andrew J.

Bioorganic & medicinal chemistry letters, 2008-02, Vol.18 (4), p.1490-1494 [Periódico revisado por pares]

Elsevier Ltd

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5
Fused tricyclic indoles as S1P1 agonists with robust efficacy in animal models of autoimmune disease
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Artigo
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Fused tricyclic indoles as S1P1 agonists with robust efficacy in animal models of autoimmune disease

Buzard, Daniel J. ; Han, Sangdon ; Lopez, Luis ; Kawasaki, Andrew ; Moody, Jeanne ; Thoresen, Lars ; Ullman, Brett ; Lehmann, Juerg ; Calderon, Imelda ; Zhu, Xiuwen ; Gharbaoui, Tawfik ; Sengupta, Dipanjan ; Krishnan, Ashwin ; Gao, Yinghong ; Edwards, Jeff ; Barden, Jeremy ; Morgan, Michael ; Usmani, Khawja ; Chen, Chuan ; Sadeque, Abu ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Liu, Ling ; Al-Shamma, Hussien ; Gatlin, Joel ; Le, Minh ; Xing, Charles ; Espinola, Sheryll ; Jones, Robert M.

Bioorganic & medicinal chemistry letters, 2012-07, Vol.22 (13), p.4404-4409 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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