Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
---|---|---|---|
1 |
Material Type: Artigo
|
Discovery and preclinical evaluations of TQB3616, a novel CDK4-biased inhibitorXu, Zhaobing ; Liu, Yingchun ; Song, Baohui ; Ren, Bingjie ; Xu, Xiongbin ; Lin, Ruibin ; Zhu, Xiaoyu ; Chen, Chen ; Yang, Shuqun ; Zhu, Yusong ; Jiang, Wen ; Li, Wei ; Xia, Yuanfeng ; Hu, Lihong ; Chen, Shuhui ; Chan, Chi-chung ; Li, Jian ; Zhang, Xiquan ; Yang, Ling ; Tian, Xin ; Ding, Charles Z.Bioorganic & medicinal chemistry letters, 2024-07, Vol.107, p.129769-129769, Article 129769 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
2 |
Material Type: Artigo
|
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido[2,3-d]pyrimidin-7-one-based SOS1 inhibitorWang, Kun ; Zhou, Zehui ; Ma, Xinyi ; Xu, Jiahang ; Xu, Wangyang ; Zhou, Guizhen ; Zhou, Chuan ; Li, Huajie ; Zheng, Mingyue ; Zhang, Sulin ; Xu, TianfengBioorganic & medicinal chemistry letters, 2024-07, Vol.107, p.129780-129780, Article 129780 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
3 |
Material Type: Artigo
|
Design, synthesis, and biological evaluation of chalcone acetamide derivatives against triple negative breast cancerKumar, Puneet ; Singh, Ruhi ; Sharma, Deepak ; Hassan, Qazi Parvaiz ; Gopu, Boobalan ; Anal, Jasha Momo H.Bioorganic & medicinal chemistry letters, 2024-07, Vol.107, p.129795-129795, Article 129795 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
4 |
Material Type: Artigo
|
Synthesis and cytotoxicity of novel 6,8,9-trisubstituted purine analogs against liver cancer cellsFatih Polat, M. ; Durmaz Şahin, Irem ; Kul, Pınar ; Cetin Atalay, Rengul ; Tuncbilek, MeralBioorganic & medicinal chemistry letters, 2024-07, Vol.106, p.129775-129775, Article 129775 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
5 |
Material Type: Artigo
|
Modification of the phenyl ring B of phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates by pyridinyl moiety leads to novel antimitotics targeting the colchicine-binding siteOuellette, Vincent ; Bouzriba, Chahrazed ; Chavez Alvarez, Atziri Corin ; Hamel-Côté, Geneviève ; Fortin, SébastienBioorganic & medicinal chemistry letters, 2024-06, Vol.105, p.129745-129745, Article 129745 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
6 |
Material Type: Artigo
|
Design, synthesis and activity evaluation of quinolinone derivatives as EZH2 inhibitorsCai, Jin ; You, Haoyuan ; Qin, Xintong ; Wang, Yuhong ; Li, WeiBioorganic & medicinal chemistry letters, 2024-06, Vol.105, p.129726-129726, Article 129726 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
7 |
Material Type: Artigo
|
Insights into the structure–activity relationship of the anticancer compound ZJ-101: A role played by the amide moietyQiu, Haibo ; Qian, Shan ; Head, Sarah A. ; Sanchez, Phillip R. ; Liu, Jun O. ; Jin, ZhendongBioorganic & medicinal chemistry letters, 2024-06, Vol.105, p.129741-129741, Article 129741 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
8 |
Material Type: Artigo
|
Identification of a novel histone H2A mono-ubiquitination-inhibiting cell-active small moleculeNi, Siyao ; Takada, Yuri ; Ando, Takaaki ; Yu, Shengwang ; Yamashita, Yasunobu ; Takahashi, Yukari ; Sawada, Miho ; Oba, Makoto ; Itoh, Yukihiro ; Suzuki, TakayoshiBioorganic & medicinal chemistry letters, 2024-06, Vol.105, p.129759-129759, Article 129759 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
9 |
Material Type: Artigo
|
Biological evaluation of sulfonate and sulfate analogues of lithocholic acid: A bioisosterism-guided approach towards the discovery of potential sialyltransferase inhibitors for antimetastatic studyPerez, Ser John Lynon P. ; Chen, Chia-Ling ; Chang, Tzu-Ting ; Li, Wen-ShanBioorganic & medicinal chemistry letters, 2024-06, Vol.105, p.129760-129760, Article 129760 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
|
10 |
Material Type: Artigo
|
Antiproliferative activities through accelerating autophagic flux by basidalin and its analogs in human cancer cellsMatagawa, Tomoe ; Sasazawa, Yukiko ; Agui, Koki ; Fujimaki, Motoki ; Kawano, Sayaka ; Ogura, Akihiro ; Takao, Ken-ichi ; Igarashi, Masayuki ; Simizu, SiroBioorganic & medicinal chemistry letters, 2024-05, Vol.104, p.129713-129713, Article 129713 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |