Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
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1 |
Material Type: Artigo
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A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptidesSun, Hongmao ; Greeley, David N. ; Chu, Xin-Jie ; Cheung, Adrian ; Danho, Waleed ; Swistok, Joseph ; Wang, Yao ; Zhao, Chunlin ; Chen, Li ; Fry, David C.Bioorganic & medicinal chemistry, 2004-05, Vol.12 (10), p.2671-2677 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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2 |
Material Type: Artigo
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Designed modification of partial agonist of ORL1 nociceptin receptor for conversion into highly potent antagonistLi, Jinglan ; Isozaki, Kaname ; Okada, Kazushi ; Matsushima, Ayami ; Nose, Takeru ; Costa, Tommaso ; Shimohigashi, YasuyukiBioorganic & medicinal chemistry, 2008-03, Vol.16 (5), p.2635-2644 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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3 |
Material Type: Artigo
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Synergistic effect of basic residues at positions 14–15 of nociceptin on binding affinity and receptor activationOkada, Kazushi ; Isozaki, Kaname ; Li, Jinglan ; Matsushima, Ayami ; Nose, Takeru ; Costa, Tommaso ; Shimohigashi, YasuyukiBioorganic & medicinal chemistry, 2008-10, Vol.16 (20), p.9261-9267 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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4 |
Material Type: Artigo
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Peptide backbone modifications on the C-terminal hexapeptide of neurotensinEinsiedel, Jürgen ; Hübner, Harald ; Hervet, Maud ; Härterich, Steffen ; Koschatzky, Susanne ; Gmeiner, PeterBioorganic & medicinal chemistry, 2008-03, Vol.18 (6), p.2013-2018 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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5 |
Material Type: Artigo
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Synthesis of a novel potent cyclic peptide MC4-ligand by ring-closing metathesisWels, Bas ; Kruijtzer, John A.W. ; Garner, Keith ; Nijenhuis, Wouter A.J. ; Gispen, Willem Hendrik ; Adan, Roger A.H. ; Liskamp, Rob M.J.Bioorganic & medicinal chemistry, 2005-07, Vol.13 (13), p.4221-4227 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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6 |
Material Type: Artigo
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ORL1 and opioid receptor preferences of nociceptin and dynorphin A analogues with Dmp substituted for N-terminal aromatic residuesSasaki, Yusuke ; Kawano, Susumu ; Kohara, Hirokazu ; Watanabe, Hideko ; Ambo, AkihiroBioorganic & medicinal chemistry, 2006-04, Vol.14 (7), p.2433-2437 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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The discovery of GSK221149A: A potent and selective oxytocin antagonistLiddle, John ; Allen, Michael J. ; Borthwick, Alan D. ; Brooks, David P. ; Davies, David E. ; Edwards, Richard M. ; Exall, Anne M. ; Hamlett, Chris ; Irving, Wendy R. ; Mason, Andrew M. ; McCafferty, Gerald P. ; Nerozzi, Fabrizio ; Peace, Simon ; Philp, Joanne ; Pollard, Derek ; Pullen, Mark A. ; Shabbir, Shaila S. ; Sollis, Steve L. ; Westfall, Timothy D. ; Woollard, Pat M. ; Wu, Charlene ; Hickey, Deirdre M.B.Bioorganic & medicinal chemistry, 2008, Vol.18 (1), p.90-94 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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8 |
Material Type: Artigo
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Synthesis and Biological Studies of Novel Neurotensin(8–13) MimeticsHong, Feng ; Zaidi, Javid ; Cusack, Bernadette ; Richelson, ElliottBioorganic & medicinal chemistry, 2002-12, Vol.10 (12), p.3849-3858 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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9 |
Material Type: Artigo
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Potent benzimidazolone-based CGRP receptor antagonistsTHEBERGE, Cory R ; BEDNAR, Rodney A ; WILLIAMS, Theresa M ; ZARTMAN, C. Blair ; ZHANG, Xu-Fang ; GRAHAM, Samuel L ; VACCA, Joseph P ; BELL, Ian M ; CORCORAN, Halea A ; FAY, John F ; HERSHEY, James C ; JOHNSTON, Victor K ; KANE, Stefanie A ; MOSSER, Scott ; SALVATORE, Christopher ABioorganic & medicinal chemistry, 2008-12, Vol.18 (23), p.6122-6125 [Periódico revisado por pares]Amsterdam: ElsevierTexto completo disponível |
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10 |
Material Type: Artigo
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Structure–activity study at positions 3 and 4 of human neuropeptide SCamarda, Valeria ; Trapella, Claudio ; Calo’, Girolamo ; Guerrini, Remo ; Rizzi, Anna ; Ruzza, Chiara ; Fiorini, Stella ; Marzola, Erika ; Reinscheid, Rainer K. ; Regoli, Domenico ; Salvadori, SeveroBioorganic & medicinal chemistry, 2008-10, Vol.16 (19), p.8841-8845 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |