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The Importance of Being Me: Magic Methyls, Methyltransferase Inhibitors, and the Discovery of Tazemetostat
The Importance of Being Me: Magic Methyls, Methyltransferase Inhibitors, and the Discovery of Tazemetostat
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The Importance of Being Me: Magic Methyls, Methyltransferase Inhibitors, and the Discovery of Tazemetostat

Kuntz, Kevin W ; Campbell, John E ; Keilhack, Heike ; Pollock, Roy M ; Knutson, Sarah K ; Porter-Scott, Margaret ; Richon, Victoria M ; Sneeringer, Chris J ; Wigle, Tim J ; Allain, Christina J ; Majer, Christina R ; Moyer, Mikel P ; Copeland, Robert A ; Chesworth, Richard

Journal of medicinal chemistry, 2016-02, Vol.59 (4), p.1556-1564 [Periódico revisado por pares]

United States: American Chemical Society

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2
Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound
Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound
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Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound

Mitchell, Lorna H. ; Drew, Allison E. ; Ribich, Scott A. ; Rioux, Nathalie ; Swinger, Kerren K. ; Jacques, Suzanne L. ; Lingaraj, Trupti ; Boriack-Sjodin, P. Ann ; Waters, Nigel J. ; Wigle, Tim J. ; Moradei, Oscar ; Jin, Lei ; Riera, Tom ; Porter-Scott, Margaret ; Moyer, Mikel P. ; Smith, Jesse J. ; Chesworth, Richard ; Copeland, Robert A.

ACS medicinal chemistry letters, 2015-06, Vol.6 (6), p.655-659 [Periódico revisado por pares]

United States: American Chemical Society

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3
Conformational Adaptation Drives Potent, Selective and Durable Inhibition of the Human Protein Methyltransferase DOT1L
Conformational Adaptation Drives Potent, Selective and Durable Inhibition of the Human Protein Methyltransferase DOT1L
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Conformational Adaptation Drives Potent, Selective and Durable Inhibition of the Human Protein Methyltransferase DOT1L

Basavapathruni, Aravind ; Jin, Lei ; Daigle, Scott R. ; Majer, Christina R. A. ; Therkelsen, Carly A. ; Wigle, Tim J. ; Kuntz, Kevin W. ; Chesworth, Richard ; Pollock, Roy M. ; Scott, Margaret P. ; Moyer, Mikel P. ; Richon, Victoria M. ; Copeland, Robert A. ; Olhava, Edward J.

Chemical biology & drug design, 2012-12, Vol.80 (6), p.971-980 [Periódico revisado por pares]

Oxford, UK: Blackwell Publishing Ltd

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4
EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity
EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity
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EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity

Campbell, John E ; Kuntz, Kevin W ; Knutson, Sarah K ; Warholic, Natalie M ; Keilhack, Heike ; Wigle, Tim J ; Raimondi, Alejandra ; Klaus, Christine R ; Rioux, Nathalie ; Yokoi, Akira ; Kawano, Satoshi ; Minoshima, Yukinori ; Choi, Hyeong-Wook ; Porter Scott, Margaret ; Waters, Nigel J ; Smith, Jesse J ; Chesworth, Richard ; Moyer, Mikel P ; Copeland, Robert A

ACS medicinal chemistry letters, 2015-05, Vol.6 (5), p.491-495 [Periódico revisado por pares]

United States: American Chemical Society

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5
Novel Oxindole Sulfonamides and Sulfamides: EPZ031686, the First Orally Bioavailable Small Molecule SMYD3 Inhibitor
Novel Oxindole Sulfonamides and Sulfamides: EPZ031686, the First Orally Bioavailable Small Molecule SMYD3 Inhibitor
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Novel Oxindole Sulfonamides and Sulfamides: EPZ031686, the First Orally Bioavailable Small Molecule SMYD3 Inhibitor

Mitchell, Lorna H ; Boriack-Sjodin, P. Ann ; Smith, Sherri ; Thomenius, Michael ; Rioux, Nathalie ; Munchhof, Michael ; Mills, James E ; Klaus, Christine ; Totman, Jennifer ; Riera, Thomas V ; Raimondi, Alejandra ; Jacques, Suzanne L ; West, Kip ; Foley, Megan ; Waters, Nigel J ; Kuntz, Kevin W ; Wigle, Tim J ; Scott, Margaret Porter ; Copeland, Robert A ; Smith, Jesse J ; Chesworth, Richard

ACS medicinal chemistry letters, 2016-02, Vol.7 (2), p.134-138 [Periódico revisado por pares]

United States: American Chemical Society

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6
A community effort in SARS‐CoV‐2 drug discovery
A community effort in SARS‐CoV‐2 drug discovery
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A community effort in SARS‐CoV‐2 drug discovery

Schimunek, Johannes ; Noé, Frank ; Olsson, Simon ; Raich, Lluís ; Winter, Robin ; Kurnikova, Maria G. ; Narangoda, Chamali H. ; Zubatyuk, Roman ; Bosko, Ivan P. ; Furs, Konstantin V. ; Karpenko, Anna D. ; Kornoushenko, Yury V. ; Shuldau, Mikita ; Yushkevich, Artsemi ; Benabderrahmane, Mohammed B. ; Bousquet‐Melou, Patrick ; Bureau, Ronan ; Charton, Beatrice ; Cirou, Bertrand C. ; Gil, Gérard ; Allen, William J. ; Sirimulla, Suman ; Antonopoulos, Nick ; Epitropakis, Nikolaos ; Krasoulis, Agamemnon ; Theodorakis, Stavros ; Medvedev, Alexander ; Popov, Petr ; Zaretckii, Mark ; Halmich, Christina ; Hochreiter, Sepp ; Widrich, Michael ; Kumar, Ashutosh ; Jain, Moksh J. ; Korablyov, Maksym ; Liu, Cheng‐Hao ; Glaab, Enrico ; Kaiser, Florian ; Schroeder, Michael ; Pugliese, Luisa ; Athanasiou, Christina ; Beccari, Andrea ; Carloni, Paolo ; Gianquinto, Eleonora ; Goßen, Jonas ; Joseph, Benjamin P. ; Kokh, Daria B. ; Kovachka, Sandra ; Manelfi, Candida ; Musiani, Francesco ; Paiardi, Giulia ; Rossetti, Giulia ; Spyrakis, Francesca ; Tsengenes, Alexandros ; Copeland, Conner ; Gaiser, Jeremiah ; Roy, Amitava ; Venkatraman, Vishwesh ; Blaschitz, Klara ; Cespugli, Marco ; Durmaz, Vedat ; Fischer, Patrick D. ; Gorgulla, Christoph ; Gruber, Karl ; Hetmann, Michael ; Kinney, Jamie E. ; Padmanabha Das, Krishna M. ; Pandita, Shreya ; Singh, Amit ; Steinkellner, Georg ; Tesseyre, Guilhem ; Wagner, Gerhard ; Wang, Zi‐Fu ; Yust, Ryan J. ; Druzhilovskiy, Dmitry S. ; Filimonov, Dmitry A. ; Pogodin, Pavel V. ; Poroikov, Vladimir ; Rudik, Anastassia V. ; Stolbov, Leonid A. ; De Rosa, Maria ; De Simone, Giada ; Gulotta, Maria R. ; Perricone, Ugo ; Casini, Arturo ; Embree, Amanda ; Voigt, Christopher A. ; Chen, Kuang‐Yu ; Jacob, Yves ; Krischuns, Tim ; Lafaye, Pierre ; Rodríguez, M. Luis ; White, Kris M. ; Fearon, Daren ; Von Delft, Frank ; Falsafi, Babak ; Ford, Bryan ; García‐Sastre, Adolfo ; Naffakh, Nadia ; Klambauer, Günter

Molecular informatics, 2024-01, Vol.43 (1), p.e202300262-n/a [Periódico revisado por pares]

Germany: Wiley Subscription Services, Inc

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