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1
The phase 3 DUO trial: duvelisib vs ofatumumab in relapsed and refractory CLL/SLL
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Artigo
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The phase 3 DUO trial: duvelisib vs ofatumumab in relapsed and refractory CLL/SLL

Flinn, Ian W. ; Hillmen, Peter ; Montillo, Marco ; Nagy, Zsolt ; Illés, Árpád ; Etienne, Gabriel ; Delgado, Julio ; Kuss, Bryone J. ; Tam, Constantine S. ; Gasztonyi, Zoltán ; Offner, Fritz ; Lunin, Scott ; Bosch, Francesco ; Davids, Matthew S. ; Lamanna, Nicole ; Jaeger, Ulrich ; Ghia, Paolo ; Cymbalista, Florence ; Portell, Craig A. ; Skarbnik, Alan P. ; Cashen, Amanda F. ; Weaver, David T. ; Kelly, Virginia M. ; Turnbull, Barry ; Stilgenbauer, Stephan

Blood, 2018-12, Vol.132 (23), p.2446-2455 [Periódico revisado por pares]

United States: Elsevier Inc

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2
The purines: Potent and versatile small molecule inhibitors and modulators of key biological targets
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Artigo
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The purines: Potent and versatile small molecule inhibitors and modulators of key biological targets

Legraverend, Michel ; Grierson, David S.

Bioorganic & medicinal chemistry, 2006-06, Vol.14 (12), p.3987-4006 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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3
Idelalisib given front-line for treatment of chronic lymphocytic leukemia causes frequent immune-mediated hepatotoxicity
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Artigo
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Idelalisib given front-line for treatment of chronic lymphocytic leukemia causes frequent immune-mediated hepatotoxicity

Lampson, Benjamin L. ; Kasar, Siddha N. ; Matos, Tiago R. ; Morgan, Elizabeth A. ; Rassenti, Laura ; Davids, Matthew S. ; Fisher, David C. ; Freedman, Arnold S. ; Jacobson, Caron A. ; Armand, Philippe ; Abramson, Jeremy S. ; Arnason, Jon E. ; Kipps, Thomas J. ; Fein, Joshua ; Fernandes, Stacey ; Hanna, John ; Ritz, Jerome ; Kim, Haesook T. ; Brown, Jennifer R.

Blood, 2016-07, Vol.128 (2), p.195-203 [Periódico revisado por pares]

United States: Elsevier Inc

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4
Design, synthesis and biological evaluation of 6-pyridylmethylaminopurines as CDK inhibitors
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Artigo
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Design, synthesis and biological evaluation of 6-pyridylmethylaminopurines as CDK inhibitors

Wilson, Stuart C. ; Atrash, Butrus ; Barlow, Clare ; Eccles, Susan ; Fischer, Peter M. ; Hayes, Angela ; Kelland, Lloyd ; Jackson, Wayne ; Jarman, Michael ; Mirza, Amin ; Moreno, Javier ; Nutley, Bernard P. ; Raynaud, Florence I. ; Sheldrake, Peter ; Walton, Mike ; Westwood, Robert ; Whittaker, Steven ; Workman, Paul ; McDonald, Edward

Bioorganic & medicinal chemistry, 2011-11, Vol.19 (22), p.6949-6965 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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5
Tanovea® for the treatment of lymphoma in dogs
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Artigo
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Tanovea® for the treatment of lymphoma in dogs

De Clercq, Erik

Biochemical pharmacology, 2018-08, Vol.154, p.265-269 [Periódico revisado por pares]

England: Elsevier Inc

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6
The phosphoinositide 3′-kinase delta inhibitor, CAL-101, inhibits B-cell receptor signaling and chemokine networks in chronic lymphocytic leukemia
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Artigo
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The phosphoinositide 3′-kinase delta inhibitor, CAL-101, inhibits B-cell receptor signaling and chemokine networks in chronic lymphocytic leukemia

Hoellenriegel, Julia ; Meadows, Sarah A. ; Sivina, Mariela ; Wierda, William G. ; Kantarjian, Hagop ; Keating, Michael J. ; Giese, Neill ; O'Brien, Susan ; Yu, Albert ; Miller, Langdon L. ; Lannutti, Brian J. ; Burger, Jan A.

Blood, 2011-09, Vol.118 (13), p.3603-3612 [Periódico revisado por pares]

Washington, DC: Elsevier Inc

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7
Clinical severity in Lesch–Nyhan disease: The role of residual enzyme and compensatory pathways
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Artigo
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Clinical severity in Lesch–Nyhan disease: The role of residual enzyme and compensatory pathways

Fu, Rong ; Sutcliffe, Diane ; Zhao, Hong ; Huang, Xinyi ; Schretlen, David J. ; Benkovic, Steve ; Jinnah, H.A.

Molecular genetics and metabolism, 2015-01, Vol.114 (1), p.55-61 [Periódico revisado por pares]

United States: Elsevier Inc

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8
The KH domain facilitates the substrate specificity and unwinding processivity of DDX43 helicase
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Artigo
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The KH domain facilitates the substrate specificity and unwinding processivity of DDX43 helicase

Yadav, Manisha ; Singh, Ravi Shankar ; Hogan, Daniel ; Vidhyasagar, Venkatasubramanian ; Yang, Shizhuo ; Chung, Ivy Yeuk Wah ; Kusalik, Anthony ; Dmitriev, Oleg Y. ; Cygler, Miroslaw ; Wu, Yuliang

The Journal of biological chemistry, 2021-01, Vol.296, p.100085-100085, Article 100085 [Periódico revisado por pares]

United States: Elsevier Inc

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9
Discovery and optimization of novel purines as potent and selective CB2 agonists
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Discovery and optimization of novel purines as potent and selective CB2 agonists

Hollinshead, Sean P. ; Astles, Peter C. ; Chambers, Mark G. ; Johnson, Michael P. ; Palmer, John ; Tidwell, Michael W.

Bioorganic & medicinal chemistry letters, 2012-08, Vol.22 (15), p.4962-4966 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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10
Comprehensive quantitative analysis of purines and pyrimidines in the human malaria parasite using ion-pairing ultra-performance liquid chromatography–mass spectrometry
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Artigo
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Comprehensive quantitative analysis of purines and pyrimidines in the human malaria parasite using ion-pairing ultra-performance liquid chromatography–mass spectrometry

Laourdakis, Christian D. ; Merino, Emilio F. ; Neilson, Andrew P. ; Cassera, Maria B.

Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2014-09, Vol.967, p.127-133 [Periódico revisado por pares]

Netherlands: Elsevier B.V

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