Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
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1 |
Material Type: Artigo
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An Aggregation Advisor for Ligand DiscoveryIrwin, John J. ; Duan, Da ; Torosyan, Hayarpi ; Doak, Allison K. ; Ziebart, Kristin T. ; Sterling, Teague ; Tumanian, Gurgen ; Shoichet, Brian K.Journal of medicinal chemistry, 2015-09, Vol.58 (17), p.7076-7087 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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2 |
Material Type: Artigo
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Adrenomedullin 2.0: Adjusting Key Levers for Metabolic StabilitySchönauer, Ria ; Els-Heindl, Sylvia ; Fischer, Jan-Patrick ; Köbberling, Johannes ; Riedl, Bernd ; Beck-Sickinger, Annette GJournal of medicinal chemistry, 2016-06, Vol.59 (12), p.5695-5705 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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3 |
Material Type: Artigo
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Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric CompoundsDrapier, Thomas ; Geubelle, Pierre ; Bouckaert, Charlotte ; Nielsen, Lise ; Laulumaa, Saara ; Goffin, Eric ; Dilly, Sébastien ; Francotte, Pierre ; Hanson, Julien ; Pochet, Lionel ; Kastrup, Jette Sandholm ; Pirotte, BernardJournal of medicinal chemistry, 2018-06, Vol.61 (12), p.5279-5291 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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4 |
Material Type: Artigo
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7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar PotencyGoffin, Eric ; Drapier, Thomas ; Larsen, Anja Probst ; Geubelle, Pierre ; Ptak, Christopher P ; Laulumaa, Saara ; Rovinskaja, Karoline ; Gilissen, Julie ; Tullio, Pascal de ; Olsen, Lars ; Frydenvang, Karla ; Pirotte, Bernard ; Hanson, Julien ; Oswald, Robert E ; Kastrup, Jette Sandholm ; Francotte, PierreJournal of medicinal chemistry, 2018-01, Vol.61 (1), p.251-264 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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5 |
Material Type: Artigo
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Beware the Receptor VariantsHanson, JulienJournal of medicinal chemistry, 2023-12, Vol.66 (23), p.15671-15673 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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6 |
Material Type: Artigo
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Metabolomics as a Challenging Approach for Medicinal Chemistry and Personalized MedicineFrédérich, Michel ; Pirotte, Bernard ; Fillet, Marianne ; de Tullio, PascalJournal of medicinal chemistry, 2016-10, Vol.59 (19), p.8649-8666 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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7 |
Material Type: Artigo
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Development of Ligands for the Super Conserved Orphan G Protein-Coupled Receptor GPR27 with Improved Efficacy and PotencyPillaiyar, Thanigaimalai ; Wozniak, Monika ; Abboud, Dayana ; Rasch, Alexander ; Liebing, Aenne-Dorothea ; Poso, Antti ; Kronenberger, Thales ; Stäubert, Claudia ; Laufer, Stefan A. ; Hanson, JulienJournal of medicinal chemistry, 2023-12, Vol.66 (24), p.17118-17137 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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8 |
Material Type: Artigo
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Toward the First Class of Suicide Inhibitors of Kallikreins Involved in Skin DiseasesTan, Xiao ; Soualmia, Feryel ; Furio, Laetitia ; Renard, Jean-François ; Kempen, Isabelle ; Qin, Lixian ; Pagano, Maurice ; Pirotte, Bernard ; El Amri, Chahrazade ; Hovnanian, Alain ; Reboud-Ravaux, MichèleJournal of medicinal chemistry, 2015-01, Vol.58 (2), p.598-612 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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9 |
Material Type: Artigo
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Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug DesignMeanwell, Nicholas AJournal of medicinal chemistry, 2018-07, Vol.61 (14), p.5822-5880 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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10 |
Material Type: Artigo
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U.S. FDA Approved Drugs from 2015–June 2020: A PerspectiveBhutani, Priyadeep ; Joshi, Gaurav ; Raja, Nivethitha ; Bachhav, Namrata ; Rajanna, Prabhakar K ; Bhutani, Hemant ; Paul, Atish T ; Kumar, RajJournal of medicinal chemistry, 2021-03, Vol.64 (5), p.2339-2381 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |