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1 |
Material Type: Artigo
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Cyclic benzamidines as orally efficacious NR2B-selective NMDA receptor antagonistsNguyen, Kevin T. ; Claiborne, Christopher F. ; McCauley, John A. ; Libby, Brian E. ; Claremon, David A. ; Bednar, Rodney A. ; Mosser, Scott D. ; Gaul, Stanley L. ; Connolly, Thomas M. ; Condra, Cindra L. ; Bednar, Bohumil ; Stump, Gary L. ; Lynch, Joseph J. ; Koblan, Kenneth S. ; Liverton, Nigel J.Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (14), p.3997-4000 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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2 |
Material Type: Artigo
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Thiourea inhibitors of herpes viruses. Part 2: N-Benzyl- N′-arylthiourea inhibitors of CMVBloom, Jonathan D. ; Dushin, Russell G. ; Curran, Kevin J. ; Donahue, Fran ; Norton, Emily B. ; Terefenko, Eugene ; Jones, Thomas R. ; Ross, Adma A. ; Feld, Boris ; Lang, Stanley A. ; DiGrandi, Martin J.Bioorganic & medicinal chemistry letters, 2004-07, Vol.14 (13), p.3401-3406 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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3 |
Material Type: Artigo
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Thiourea inhibitors of herpes viruses. part 1: bis-(aryl)thiourea inhibitors of CMVBloom, Jonathan D. ; DiGrandi, Martin J. ; Dushin, Russell G. ; Curran, Kevin J. ; Ross, Adma A. ; Norton, Emily B. ; Terefenko, Eugene ; Jones, Thomas R. ; Feld, Boris ; Lang, Stanley A.Bioorganic & medicinal chemistry letters, 2003-09, Vol.13 (17), p.2929-2932 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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4 |
Material Type: Artigo
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Orally Efficacious NR2B-Selective NMDA Receptor AntagonistsClaiborne, Christopher F ; McCauley, John A ; Libby, Brian E ; Curtis, Neil R ; Diggle, Helen J ; Kulagowski, Janusz J ; Michelson, Stuart R ; Anderson, Kenneth D ; Claremon, David A ; Freidinger, Roger M ; Bednar, Rodney A ; Mosser, Scott D ; Gaul, Stanley L ; Connolly, Thomas M ; Condra, Cindra L ; Bednar, Bohumil ; Stump, Gary L ; Lynch, Joseph J ; Macaulay, Alison ; Wafford, Keith A ; Koblan, Kenneth S ; Liverton, Nigel JBioorganic & medicinal chemistry letters, 2003-02, Vol.13 (4), p.697-700 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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5 |
Material Type: Artigo
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Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2- d]pyrimidines as EGFR and ErbB-2 inhibitorsStevens, Kirk L. ; Alligood, Krystal J. ; Alberti, Jennifer G. Badiang ; Caferro, Thomas R. ; Chamberlain, Stanley D. ; Dickerson, Scott H. ; Dickson, Hamilton D. ; Emerson, Holly K. ; Griffin, Robert J. ; Hubbard, Robert D. ; Keith, Barry R. ; Mullin, Robert J. ; Petrov, Kimberly G. ; Gerding, Roseanne M. ; Reno, Michael J. ; Rheault, Tara R. ; Rusnak, David W. ; Sammond, Douglas M. ; Smith, Stephon C. ; Uehling, David E. ; Waterson, Alex G. ; Wood, Edgar R.Bioorganic & medicinal chemistry letters, 2009, Vol.19 (1), p.21-26 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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6 |
Material Type: Artigo
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Novel, potent and selective cyclin D1/CDK4 inhibitors: indolo[6,7- a]pyrrolo[3,4- c]carbazolesEngler, Thomas A. ; Furness, Kelly ; Malhotra, Sushant ; Sanchez-Martinez, Concha ; Shih, Chuan ; Xie, Walter ; Zhu, Guoxin ; Zhou, Xun ; Conner, Scott ; Faul, Margaret M. ; Sullivan, Kevin A. ; Kolis, Stanley P. ; Brooks, Harold B. ; Patel, Bharvin ; Schultz, Richard M. ; DeHahn, Tammy B. ; Kirmani, Kashif ; Spencer, Charles D. ; Watkins, Scott A. ; Considine, Eileen L. ; Dempsey, Jack A. ; Ogg, Catherine A. ; Stamm, Nancy B. ; Anderson, Bryan D. ; Campbell, Robert M. ; Vasudevan, Vasu ; Lytle, Michelle L.Bioorganic & medicinal chemistry letters, 2003-07, Vol.13 (14), p.2261-2267 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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Discovery of a nonpeptidic small molecule antagonist of the human platelet thrombin receptor (PAR-1)Nantermet, Philippe G ; Barrow, James C ; Lundell, George F ; Pellicore, Janetta M ; Rittle, Kenneth E ; Young, MaryBeth ; Freidinger, Roger M ; Connolly, Thomas M ; Condra, Cindra ; Karczewski, Jerzy ; Bednar, Rodney A ; Gaul, Stanley L ; Gould, Robert J ; Prendergast, Kris ; Selnick, Harold GBioorganic & medicinal chemistry letters, 2002-02, Vol.12 (3), p.319-323 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |