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1
The expanding reaction toolkit for DNA-encoded libraries
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The expanding reaction toolkit for DNA-encoded libraries

Fair, Richard J. ; Walsh, Ryan T. ; Hupp, Christopher D.

Bioorganic & medicinal chemistry letters, 2021-11, Vol.51, p.128339-128339, Article 128339 [Periódico revisado por pares]

England: Elsevier Ltd

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2
Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry
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Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry

Mondal, Milon ; Radeva, Nedyalka ; Fanlo-Virgós, Hugo ; Otto, Sijbren ; Klebe, Gerhard ; Hirsch, Anna K. H.

Angewandte Chemie (International ed.), 2016-08, Vol.55 (32), p.9422-9426 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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3
Bio-instructive materials on-demand - combinatorial chemistry of peptoids, foldamers, and beyond
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Bio-instructive materials on-demand - combinatorial chemistry of peptoids, foldamers, and beyond

Herlan, Claudine Nicole ; Feser, Dominik ; Schepers, Ute ; Bräse, Stefan

Chemical communications (Cambridge, England), 2021-10, Vol.57 (85), p.11131-11152 [Periódico revisado por pares]

England: Royal Society of Chemistry

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4
Analysis of Current DNA Encoded Library Screening Data Indicates Higher False Negative Rates for Numerically Larger Libraries
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Analysis of Current DNA Encoded Library Screening Data Indicates Higher False Negative Rates for Numerically Larger Libraries

Satz, Alexander L ; Hochstrasser, Remo ; Petersen, Ann C

ACS combinatorial science, 2017-04, Vol.19 (4), p.234-238 [Periódico revisado por pares]

United States: American Chemical Society

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5
Strategies for Heterocyclic Construction via Novel Multicomponent Reactions Based on Isocyanides and Nucleophilic Carbenes
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Strategies for Heterocyclic Construction via Novel Multicomponent Reactions Based on Isocyanides and Nucleophilic Carbenes

Nair, Vijay ; Rajesh, C ; Vinod, A. U ; Bindu, S ; Sreekanth, A. R ; Mathen, J. S ; Balagopal, Lakshmi

Accounts of chemical research, 2003-12, Vol.36 (12), p.899-907 [Periódico revisado por pares]

United States: American Chemical Society

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6
Current Parallel Solid-Phase Synthesis of Drug-like Oxadiazole and Thiadiazole Derivatives for Combinatorial Chemistry
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Current Parallel Solid-Phase Synthesis of Drug-like Oxadiazole and Thiadiazole Derivatives for Combinatorial Chemistry

Abdildinova, Aizhan ; Gong, Young-Dae

ACS combinatorial science, 2018-06, Vol.20 (6), p.309-329 [Periódico revisado por pares]

United States: American Chemical Society

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7
Identification and synthesis of an efficient multivalent E. coli heat labile toxin inhibitor __ A dynamic combinatorial chemistry approach
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Identification and synthesis of an efficient multivalent E. coli heat labile toxin inhibitor __ A dynamic combinatorial chemistry approach

Xu, Jintao ; Zhang, Shixin ; Zhao, Shuang ; Hu, Lei

Bioorganic & medicinal chemistry, 2020-05, Vol.28 (9), p.115436-115436, Article 115436 [Periódico revisado por pares]

England: Elsevier Ltd

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8
Synthesis of Heterocycles by Formal Cycloadditions of Isocyanides
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Synthesis of Heterocycles by Formal Cycloadditions of Isocyanides

Kruithof, Art ; Ruijter, Eelco ; Orru, Romano V. A.

Chemistry, an Asian journal, 2015-03, Vol.10 (3), p.508-520 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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9
Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase
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Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase

Ortiz, Maria A. ; Michaels, Heather ; Molina, Brandon ; Toenjes, Sean ; Davis, Jennifer ; Marconi, Guya Diletta ; Hecht, David ; Gustafson, Jeffrey L. ; Piedrafita, F. Javier ; Nefzi, Adel

Bioorganic & medicinal chemistry letters, 2020-05, Vol.30 (9), p.127108-127108, Article 127108 [Periódico revisado por pares]

England: Elsevier Ltd

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10
Salt-Induced Adaptation of a Dynamic Combinatorial Library of Pseudopeptidic Macrocycles: Unraveling the Electrostatic Effects in Mixed Aqueous Media
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Salt-Induced Adaptation of a Dynamic Combinatorial Library of Pseudopeptidic Macrocycles: Unraveling the Electrostatic Effects in Mixed Aqueous Media

Atcher, Joan ; Moure, Alejandra ; Bujons, Jordi ; Alfonso, Ignacio

Chemistry : a European journal, 2015-04, Vol.21 (18), p.6869-6878 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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