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11 |
Material Type: Artigo
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Development of matrix metalloproteinase-13 inhibitors – A structure-activity/structure-property relationship studyFuerst, Rita ; Yong Choi, Jun ; Knapinska, Anna M. ; Smith, Lyndsay ; Cameron, Michael D. ; Ruiz, Claudia ; Fields, Gregg B. ; Roush, William R.Bioorganic & medicinal chemistry, 2018-10, Vol.26 (18), p.4984-4995 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
12 |
Material Type: Artigo
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A panoramic review of IL-6: Structure, pathophysiological roles and inhibitorsKaur, Sukhvir ; Bansal, Yogita ; Kumar, Raj ; Bansal, GulshanBioorganic & medicinal chemistry, 2020-03, Vol.28 (5), p.115327-115327, Article 115327 [Periódico revisado por pares]EnglandTexto completo disponível |
13 |
Material Type: Artigo
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Targeting zoonotic viruses: Structure-based inhibition of the 3C-like protease from bat coronavirus HKU4—The likely reservoir host to the human coronavirus that causes Middle East Respiratory Syndrome (MERS)St. John, Sarah E. ; Tomar, Sakshi ; Stauffer, Shaun R. ; Mesecar, Andrew D.Bioorganic & medicinal chemistry, 2015-09, Vol.23 (17), p.6036-6048 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
14 |
Material Type: Artigo
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Synthesis and evaluation of pharmacological profile of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1 H)-sulfonamidesGitto, Rosaria ; Ferro, Stefania ; Agnello, Stefano ; De Luca, Laura ; De Sarro, Giovanbattista ; Russo, Emilio ; Vullo, Daniela ; Supuran, Claudiu T. ; Chimirri, AlbaBioorganic & medicinal chemistry, 2009-05, Vol.17 (10), p.3659-3664 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
15 |
Material Type: Artigo
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Design and synthesis of a potent inhibitor of class 1 DYRK kinases as a suppressor of adipogenesisMasaki, So ; Kii, Isao ; Sumida, Yuto ; Kato-Sumida, Tomoe ; Ogawa, Yasushi ; Ito, Nobutoshi ; Nakamura, Mitsuhiro ; Sonamoto, Rie ; Kataoka, Naoyuki ; Hosoya, Takamitsu ; Hagiwara, MasatoshiBioorganic & medicinal chemistry, 2015-08, Vol.23 (15), p.4434-4441 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
16 |
Material Type: Artigo
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Synthesis of novel indole-thiazolidinone hybrid structures as promising scaffold with anticancer potentialKryshchyshyn-Dylevych, Anna ; Radko, Lidia ; Finiuk, Nataliya ; Garazd, Myroslav ; Kashchak, Nataliya ; Posyniak, Andrzej ; Niemczuk, Krzysztof ; Stoika, Rostyslav ; Lesyk, RomanBioorganic & medicinal chemistry, 2021-11, Vol.50, p.116453, Article 116453 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
17 |
Material Type: Artigo
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Structure, function and applications of carbonic anhydrase isozymesImtaiyaz Hassan, Md ; Shajee, Bushra ; Waheed, Abdul ; Ahmad, Faizan ; Sly, William S.Bioorganic & medicinal chemistry, 2013-03, Vol.21 (6), p.1570-1582 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
18 |
Material Type: Artigo
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Synthesis and structure-activity relationships for new 6-fluoroquinoline derivatives with antiplasmodial activityHochegger, Patrick ; Faist, Johanna ; Seebacher, Werner ; Saf, Robert ; Mäser, Pascal ; Kaiser, Marcel ; Weis, RobertBioorganic & medicinal chemistry, 2019-05, Vol.27 (10), p.2052-2065 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
19 |
Material Type: Artigo
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The structure–activity relationship of urea derivatives as anti-tuberculosis agentsBrown, Joshua R. ; North, Elton J. ; Hurdle, Julian G. ; Morisseau, Christophe ; Scarborough, Jerrod S. ; Sun, Dianqing ; Korduláková, Jana ; Scherman, Michael S. ; Jones, Victoria ; Grzegorzewicz, Anna ; Crew, Rebecca M. ; Jackson, Mary ; McNeil, Michael R. ; Lee, Richard E.Bioorganic & medicinal chemistry, 2011-09, Vol.19 (18), p.5585-5595 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
20 |
Material Type: Artigo
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Inhibitors of protein arginine deiminases and their efficacy in animal models of multiple sclerosisSarswat, Amit ; Wasilewski, Ewa ; Chakka, Sai K. ; Bello, Angelica M. ; Caprariello, Andrew V. ; Muthuramu, Chithra M. ; Stys, Peter K. ; Dunn, Shannon E. ; Kotra, Lakshmi P.Bioorganic & medicinal chemistry, 2017-05, Vol.25 (9), p.2643-2656 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |