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1
Process Research and Development and Scale-up of a 4,4-Difluoro-3,3-dimethylproline Derivative
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Artigo
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Process Research and Development and Scale-up of a 4,4-Difluoro-3,3-dimethylproline Derivative

Rossi, Francesco ; Corcella, Francesco ; Caldarelli, Francesco Saverio ; Heidempergher, Franco ; Marchionni, Chiara ; Auguadro, Miriam ; Cattaneo, Marco ; Ceriani, Lucio ; Visentin, Giuseppina ; Ventrella, Giambattista ; Pinciroli, Vittorio ; Ramella, Giuliano ; Candiani, Ilaria ; Bedeschi, Angelo ; Tomasi, Attilio ; Kline, Billie J ; Martinez, Carlos A ; Yazbeck, Daniel ; Kucera, David J

Organic process research & development, 2008-03, Vol.12 (2), p.322-338 [Periódico revisado por pares]

American Chemical Society

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2
Synthesis and Anticonvulsant Activity of a New Class of 2-[(Arylalkyl)amino]alkanamide Derivatives
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Artigo
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Synthesis and Anticonvulsant Activity of a New Class of 2-[(Arylalkyl)amino]alkanamide Derivatives

Pevarello, Paolo ; Bonsignori, Alberto ; Dostert, Philippe ; Heidempergher, Franco ; Pinciroli, Vittorio ; Colombo, Maristella ; McArthur, Robert A ; Salvati, Patricia ; Post, Claes ; Fariello, Ruggero G ; Varasi, Mario

Journal of medicinal chemistry, 1998-02, Vol.41 (4), p.579-590 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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3
Development of Scaffold Synthesis for the Preparation of New Insulin-Like Growth Factor 1 Receptor Inhibitors
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Artigo
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Development of Scaffold Synthesis for the Preparation of New Insulin-Like Growth Factor 1 Receptor Inhibitors

Candiani, Ilaria ; D’Arasmo, Germano ; Heidempergher, Franco ; Tomasi, Attilio

Organic process research & development, 2009-05, Vol.13 (3), p.456-462 [Periódico revisado por pares]

American Chemical Society

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4
Phenylimidazolidin-2-one Derivatives as Selective 5-HT3 Receptor Antagonists and Refinement of the Pharmacophore Model for 5-HT3 Receptor Binding
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Artigo
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Phenylimidazolidin-2-one Derivatives as Selective 5-HT3 Receptor Antagonists and Refinement of the Pharmacophore Model for 5-HT3 Receptor Binding

Heidempergher, Franco ; Pillan, Antonio ; Pinciroli, Vittorio ; Vaghi, Fabrizio ; Arrigoni, Claudio ; Bolis, Giorgio ; Caccia, Carla ; Dho, Luciano ; McArthur, Robert ; Varasi, Mario

Journal of medicinal chemistry, 1997-10, Vol.40 (21), p.3369-3380 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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5
Phenylimidazolidin-2-one Derivatives as Selective 5-HT 3 Receptor Antagonists and Refinement of the Pharmacophore Model for 5-HT 3 Receptor Binding
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Artigo
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Phenylimidazolidin-2-one Derivatives as Selective 5-HT 3 Receptor Antagonists and Refinement of the Pharmacophore Model for 5-HT 3 Receptor Binding

Heidempergher, Franco ; Pillan, Antonio ; Pinciroli, Vittorio ; Vaghi, Fabrizio ; Arrigoni, Claudio ; Bolis, Giorgio ; Caccia, Carla ; Dho, Luciano ; McArthur, Robert ; Varasi, Mario

Journal of medicinal chemistry, 1997-10, Vol.40 (21), p.3369-3380 [Periódico revisado por pares]

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6
Pyrrolo[3,2- c]quinoline derivatives: a new class of kynurenine-3-hydroxylase inhibitors
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Artigo
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Pyrrolo[3,2- c]quinoline derivatives: a new class of kynurenine-3-hydroxylase inhibitors

Heidempergher, Franco ; Pevarello, Paolo ; Pillan, Antonio ; Pinciroli, Vittorio ; Della Torre, Arturo ; Speciale, Carmela ; Marconi, Marina ; Cini, Massimo ; Toma, Salvatore ; Greco, Felicita ; Varasi, Mario

Farmaco (Società chimica italiana : 1989), 1999-03, Vol.54 (3), p.152-160 [Periódico revisado por pares]

Lausanne: Elsevier SAS

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7
Preparation of 7-oxaaporphine derivatives and evaluation of their dopaminergic activity
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Artigo
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Preparation of 7-oxaaporphine derivatives and evaluation of their dopaminergic activity

Banzatti, Carlo ; Carfagna, Nicola ; Commisso, Roberto ; Heidempergher, Franco ; Pegrassi, Lorenzo ; Melloni, Piero

Journal of medicinal chemistry, 1988-07, Vol.31 (7), p.1466-1471 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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8
Synthesis of phenyl-substituted 2H-3,4-dihydro-3-aminomethyl-1,4-benzoxazines. Intermediates for 1H-2,3,3a,4-tetrahydroimidazo[5,1-c][1,4]benzoxazin-1-one derivatives. Part II
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Artigo
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Synthesis of phenyl-substituted 2H-3,4-dihydro-3-aminomethyl-1,4-benzoxazines. Intermediates for 1H-2,3,3a,4-tetrahydroimidazo[5,1-c][1,4]benzoxazin-1-one derivatives. Part II

Banzatti, Carlo ; Heidempergher, Franco ; Melloni, Piero

Journal of heterocyclic chemistry, 1983-03, Vol.20 (2), p.259-265 [Periódico revisado por pares]

Hoboken: Wiley-Blackwell

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9
Synthesis of phenyl‐substituted 2 H ‐3,4‐dihydro‐3‐aminomethyl‐1,4‐benzoxazines. Intermediates for 1 H ‐2,3,3a,4‐tetrahydroimidazo[5,1‐ c ][1,4]benzoxazin‐1‐one derivatives. Part II
Material Type:
Artigo
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Synthesis of phenyl‐substituted 2 H ‐3,4‐dihydro‐3‐aminomethyl‐1,4‐benzoxazines. Intermediates for 1 H ‐2,3,3a,4‐tetrahydroimidazo[5,1‐ c ][1,4]benzoxazin‐1‐one derivatives. Part II

Banzatti, Carlo ; Heidempergher, Franco ; Melloni, Piero

Journal of heterocyclic chemistry, 1983-03, Vol.20 (2), p.259-265 [Periódico revisado por pares]

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