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Material Type: Artigo
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α‑Ketoamides as Broad-Spectrum Inhibitors of Coronavirus and Enterovirus Replication: Structure-Based Design, Synthesis, and Activity AssessmentZhang, Linlin ; Lin, Daizong ; Kusov, Yuri ; Nian, Yong ; Ma, Qingjun ; Wang, Jiang ; von Brunn, Albrecht ; Leyssen, Pieter ; Lanko, Kristina ; Neyts, Johan ; de Wilde, Adriaan ; Snijder, Eric J ; Liu, Hong ; Hilgenfeld, RolfJournal of medicinal chemistry, 2020-05, Vol.63 (9), p.4562-4578 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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2 |
Material Type: Artigo
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Isoxazolidine: A Privileged Scaffold for Organic and Medicinal ChemistryBerthet, Mathéo ; Cheviet, Thomas ; Dujardin, Gilles ; Parrot, Isabelle ; Martinez, JeanChemical reviews, 2016-12, Vol.116 (24), p.15235-15283 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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3 |
Material Type: Artigo
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2,5-Diketopiperazines: Synthesis, Reactions, Medicinal Chemistry, and Bioactive Natural ProductsBorthwick, Alan DChemical reviews, 2012-07, Vol.112 (7), p.3641-3716 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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4 |
Material Type: Artigo
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Poly(2‐Oxazoline)‐Based Functional Peptide Mimics: Eradicating MRSA Infections and Persisters while Alleviating Antimicrobial ResistanceZhou, Min ; Qian, Yuxin ; Xie, Jiayang ; Zhang, Wenjing ; Jiang, Weinan ; Xiao, Ximian ; Chen, Sheng ; Dai, Chengzhi ; Cong, Zihao ; Ji, Zhemin ; Shao, Ning ; Liu, Longqiang ; Wu, Yuequn ; Liu, RunhuiAngewandte Chemie (International ed.), 2020-04, Vol.59 (16), p.6412-6419 [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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5 |
Material Type: Artigo
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3CL Protease Inhibitors with an Electrophilic Arylketone Moiety as Anti-SARS-CoV‑2 AgentsKonno, Sho ; Kobayashi, Kiyotaka ; Senda, Miki ; Funai, Yuta ; Seki, Yuta ; Tamai, Ikumi ; Schäkel, Laura ; Sakata, Kyousuke ; Pillaiyar, Thanigaimalai ; Taguchi, Akihiro ; Taniguchi, Atsuhiko ; Gütschow, Michael ; Müller, Christa E ; Takeuchi, Koh ; Hirohama, Mikako ; Kawaguchi, Atsushi ; Kojima, Masaki ; Senda, Toshiya ; Shirasaka, Yoshiyuki ; Kamitani, Wataru ; Hayashi, YoshioJournal of medicinal chemistry, 2022-02, Vol.65 (4), p.2926-2939 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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6 |
Material Type: Artigo
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Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV‑2Dai, Wenhao ; Jochmans, Dirk ; Xie, Hang ; Yang, Hang ; Li, Jian ; Su, Haixia ; Chang, Di ; Wang, Jiang ; Peng, Jingjing ; Zhu, Lili ; Nian, Yong ; Hilgenfeld, Rolf ; Jiang, Hualiang ; Chen, Kaixian ; Zhang, Leike ; Xu, Yechun ; Neyts, Johan ; Liu, HongJournal of medicinal chemistry, 2022-02, Vol.65 (4), p.2794-2808 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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7 |
Material Type: Artigo
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Hydrogen-Bonding-Driven 3D Supramolecular Assembly of Peptidomimetic ZipperTeng, Peng ; Niu, Zheng ; She, Fengyu ; Zhou, Mi ; Sang, Peng ; Gray, Geoffrey M ; Verma, Gaurav ; Wojtas, Lukasz ; van der Vaart, Arjan ; Ma, Shengqian ; Cai, JianfengJournal of the American Chemical Society, 2018-05, Vol.140 (17), p.5661-5665 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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8 |
Material Type: Artigo
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Advances in Development of Antimicrobial Peptidomimetics as Potential DrugsMolchanova, Natalia ; Hansen, Paul R ; Franzyk, HenrikMolecules (Basel, Switzerland), 2017-08, Vol.22 (9), p.1430 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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9 |
Material Type: Artigo
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Chemical Modifications Designed to Improve Peptide Stability: Incorporation of Non-Natural Amino Acids, Pseudo-Peptide Bonds, and CyclizationGentilucci, Luca ; De Marco, Rossella ; Cerisoli, LuciaCurrent pharmaceutical design, 2010-01, Vol.16 (28), p.3185-3203 [Periódico revisado por pares]United Arab Emirates: Bentham Science Publishers LtdTexto completo disponível |
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10 |
Material Type: Artigo
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Modular Design of Membrane-Active Antibiotics: From Macromolecular Antimicrobials to Small Scorpionlike PeptidomimeticsWang, Minghui ; Feng, Xiaoqian ; Gao, Ruixuan ; Sang, Peng ; Pan, Xin ; Wei, Lulu ; Lu, Chao ; Wu, Chuanbin ; Cai, JianfengJournal of medicinal chemistry, 2021-07, Vol.64 (14), p.9894-9905 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |