Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
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1 |
Material Type: Artigo
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Straightforward conversion of decoquinate into inexpensive tractable new derivatives with significant antimalarial activitiesBeteck, Richard M. ; Coertzen, Dina ; Smit, Frans J. ; Birkholtz, Lyn-Marie ; Haynes, Richard K. ; N’Da, David D.Bioorganic & medicinal chemistry letters, 2016-07, Vol.26 (13), p.3006-3009 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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2 |
Material Type: Artigo
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An orally available, brain-penetrant CAMKK2 inhibitor reduces food intake in rodent modelPrice, Daniel J. ; Drewry, David H. ; Schaller, Lee T. ; Thompson, Brian D. ; Reid, Paul R. ; Maloney, Patrick R. ; Liang, Xi ; Banker, Periette ; Buckholz, Richard G. ; Selley, Paula K. ; McDonald, Octerloney B. ; Smith, Jeffery L. ; Shearer, Todd W. ; Cox, Richard F. ; Williams, Shawn P. ; Reid, Robert A. ; Tacconi, Stefano ; Faggioni, Federico ; Piubelli, Chiara ; Sartori, Ilaria ; Tessari, Michela ; Wang, Tony Y.Bioorganic & medicinal chemistry letters, 2018-06, Vol.28 (10), p.1958-1963 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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3 |
Material Type: Artigo
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Toward the development of potent and selective bisubstrate inhibitors of protein arginine methyltransferasesDowden, James ; Hong, Wei ; Parry, Richard V. ; Pike, Richard A. ; Ward, Stephen G.Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (7), p.2103-2105 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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4 |
Material Type: Artigo
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The expanding reaction toolkit for DNA-encoded librariesFair, Richard J. ; Walsh, Ryan T. ; Hupp, Christopher D.Bioorganic & medicinal chemistry letters, 2021-11, Vol.51, p.128339-128339, Article 128339 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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5 |
Material Type: Artigo
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Pterin–sulfa conjugates as dihydropteroate synthase inhibitors and antibacterial agentsZhao, Ying ; Shadrick, William R. ; Wallace, Miranda J. ; Wu, Yinan ; Griffith, Elizabeth C. ; Qi, Jianjun ; Yun, Mi-Kyung ; White, Stephen W. ; Lee, Richard E.Bioorganic & medicinal chemistry letters, 2016-08, Vol.26 (16), p.3950-3954 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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6 |
Material Type: Artigo
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Discovery of ethyl ketone-based HDACs 1, 2, and 3 selective inhibitors for HIV latency reactivationYu, Wensheng ; Liu, Jian ; Yu, Younong ; Zhang, Vivian ; Clausen, Dane ; Kelly, Joseph ; Wolkenberg, Scott ; Beshore, Douglas ; Duffy, Joseph L. ; Chung, Christine C. ; Myers, Robert W. ; Klein, Daniel J. ; Fells, James ; Holloway, Kate ; Wu, Jin ; Wu, Guoxin ; Howell, Bonnie J. ; Barnard, Richard J.O. ; Kozlowski, JosephBioorganic & medicinal chemistry letters, 2020-07, Vol.30 (13), p.127197-127197, Article 127197 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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Optimization of novel nipecotic bis(amide) inhibitors of the Rho/MKL1/SRF transcriptional pathway as potential anti-metastasis agentsBell, Jessica L. ; Haak, Andrew J. ; Wade, Susan M. ; Kirchhoff, Paul D. ; Neubig, Richard R. ; Larsen, Scott D.Bioorganic & medicinal chemistry letters, 2013-07, Vol.23 (13), p.3826-3832 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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8 |
Material Type: Artigo
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Discovery of PH-797804, a highly selective and potent inhibitor of p38 MAP kinaseSelness, Shaun R ; Devraj, Rajesh V ; Devadas, Balekudru ; Walker, John K ; Boehm, Terri L ; Durley, Richard C ; Shieh, Huey ; Xing, Li ; Rucker, Paul V ; Jerome, Kevin D ; Benson, Alan G ; Marrufo, Laura D ; Madsen, Heather M ; Hitchcock, Jeff ; Owen, Tom J ; Christie, Lance ; Promo, Michele A ; Hickory, Brian S ; Alvira, Edgardo ; Naing, Win ; Blevis-Bal, Radhika ; Messing, Dean ; Yang, Jerry ; Mao, Michael K ; Yalamanchili, Gopi ; Vonder Embse, Richard ; Hirsch, Jeffrey ; Saabye, Matthew ; Bonar, Sheri ; Webb, Elizabeth ; Anderson, Gary ; Monahan, Joseph BBioorganic & medicinal chemistry letters, 2011-07, Vol.21 (13), p.4066-4071 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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9 |
Material Type: Artigo
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Perfluoroarene-based peptide macrocycles that inhibit the Nrf2/Keap1 interactionSteel, Richard J. ; O'Connell, Maria A. ; Searcey, MarkBioorganic & medicinal chemistry letters, 2018-09, Vol.28 (16), p.2728-2731 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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10 |
Material Type: Artigo
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Deuteration and fluorination of 1,3-bis(2-phenylethyl)pyrimidine-2,4,6(1H,3H,5H)-trione to improve its pharmacokinetic propertiesXia, Guoyao ; Benmohamed, Radhia ; Morimoto, Richard I. ; Kirsch, Donald R. ; Silverman, Richard B.Bioorganic & medicinal chemistry letters, 2014-11, Vol.24 (21), p.5098-5101 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |