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1
Design, synthesis, and biological evaluation of substituted hydrazone and pyrazole derivatives as selective COX-2 inhibitors: Molecular docking study
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Design, synthesis, and biological evaluation of substituted hydrazone and pyrazole derivatives as selective COX-2 inhibitors: Molecular docking study

El-Sayed, Magda A.-A. ; Abdel-Aziz, Naglaa I. ; Abdel-Aziz, Alaa A.-M. ; El-Azab, Adel S. ; Asiri, Yousif A. ; ElTahir, Kamal E.H.

Bioorganic & medicinal chemistry, 2011-06, Vol.19 (11), p.3416-3424 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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2
Synthesis, biological evaluation and molecular modeling study of pyrazole and pyrazoline derivatives as selective COX-2 inhibitors and anti-inflammatory agents. Part 2
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Synthesis, biological evaluation and molecular modeling study of pyrazole and pyrazoline derivatives as selective COX-2 inhibitors and anti-inflammatory agents. Part 2

El-Sayed, Magda A.-A. ; Abdel-Aziz, Naglaa I. ; Abdel-Aziz, Alaa A.-M. ; El-Azab, Adel S. ; ElTahir, Kamal E.H.

Bioorganic & medicinal chemistry, 2012-05, Vol.20 (10), p.3306-3316 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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3
Design, Synthesis and Anticancer Evaluation of New Substituted Thiophene-Quinoline Derivatives
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Design, Synthesis and Anticancer Evaluation of New Substituted Thiophene-Quinoline Derivatives

Othman, Dina I.A. ; Selim, Khalid B. ; El-Sayed, Magda A.-A. ; Tantawy, Atif S. ; Amen, Yhiya ; Shimizu, Kuniyoshi ; Okauchi, Tatsuo ; Kitamura, Mitsuru

Bioorganic & medicinal chemistry, 2019-10, Vol.27 (19), p.115026-115026, Article 115026 [Periódico revisado por pares]

England: Elsevier Ltd

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4
Synthesis and biological evaluation of 2-styrylquinolines as antitumour agents and EGFR kinase inhibitors: molecular docking study
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Synthesis and biological evaluation of 2-styrylquinolines as antitumour agents and EGFR kinase inhibitors: molecular docking study

El-Sayed, Magda A.-A. ; El-Husseiny, Walaa M. ; Abdel-Aziz, Naglaa I. ; El-Azab, Adel S. ; Abuelizz, Hatem A. ; Abdel-Aziz, Alaa A.-M.

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.199-209 [Periódico revisado por pares]

England: Taylor & Francis

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5
Synthesis, anticancer and antimicrobial evaluation of new benzofuran based derivatives: PI3K inhibition, quorum sensing and molecular modeling study
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Synthesis, anticancer and antimicrobial evaluation of new benzofuran based derivatives: PI3K inhibition, quorum sensing and molecular modeling study

El-Khouly, Omar A. ; Henen, Morkos A. ; El-Sayed, Magda A.-A. ; Shabaan, Mona I. ; El-Messery, Shahenda M.

Bioorganic & medicinal chemistry, 2021-02, Vol.31, p.115976-115976, Article 115976 [Periódico revisado por pares]

England: Elsevier Ltd

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6
Synthesis, antitumor activity and molecular docking study of some novel 3-benzyl-4(3H)quinazolinone analogues
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Synthesis, antitumor activity and molecular docking study of some novel 3-benzyl-4(3H)quinazolinone analogues

Al-Suwaidan, Ibrahim A. ; Abdel-Aziz, Alaa A.-M. ; Shawer, Taghreed Z. ; Ayyad, Rezk R. ; Alanazi, Amer M. ; El-Morsy, Ahmad M. ; Mohamed, Menshawy A. ; Abdel-Aziz, Naglaa I. ; El-Sayed, Magda A.-A. ; El-Azab, Adel S.

Journal of enzyme inhibition and medicinal chemistry, 2016-01, Vol.31 (1), p.78-89 [Periódico revisado por pares]

England: Taylor & Francis

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7
Synthesis, antitumour and antioxidant activities of novel α,β-unsaturated ketones and related heterocyclic analogues: EGFR inhibition and molecular modelling study
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Synthesis, antitumour and antioxidant activities of novel α,β-unsaturated ketones and related heterocyclic analogues: EGFR inhibition and molecular modelling study

El-Husseiny, Walaa M. ; El-Sayed, Magda A.-A. ; Abdel-Aziz, Naglaa I. ; El-Azab, Adel S. ; Ahmed, Esam R. ; Abdel-Aziz, Alaa A.-M.

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.507-518 [Periódico revisado por pares]

England: Taylor & Francis

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8
Synthesis, antitumor activity, and molecular docking study of 2-cyclopentyloxyanisole derivatives: mechanistic study of enzyme inhibition
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Synthesis, antitumor activity, and molecular docking study of 2-cyclopentyloxyanisole derivatives: mechanistic study of enzyme inhibition

El-Husseiny, Walaa M. ; El-Sayed, Magda A.-A. ; El-Azab, Adel S. ; AlSaif, Nawaf A. ; Alanazi, Mohammed M. ; Abdel-Aziz, Alaa A.-M.

Journal of enzyme inhibition and medicinal chemistry, 2020-01, Vol.35 (1), p.744-758 [Periódico revisado por pares]

England: Taylor & Francis

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9
Synthesis, antitumour activities and molecular docking of thiocarboxylic acid ester-based NSAID scaffolds: COX-2 inhibition and mechanistic studies
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Synthesis, antitumour activities and molecular docking of thiocarboxylic acid ester-based NSAID scaffolds: COX-2 inhibition and mechanistic studies

El-Azab, Adel S. ; Abdel-Aziz, Alaa A.-M. ; Abou-Zeid, Laila A. ; El-Husseiny, Walaa M. ; El_Morsy, Ahmad M. ; El-Gendy, Manal A. ; El-Sayed, Magda A.-A.

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.989-998 [Periódico revisado por pares]

England: Taylor & Francis

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10
In vitro cytotoxicity and docking study of novel symmetric and asymmetric dihydropyridines and pyridines as EGFR tyrosine kinase inhibitors
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In vitro cytotoxicity and docking study of novel symmetric and asymmetric dihydropyridines and pyridines as EGFR tyrosine kinase inhibitors

Mansour, Basem ; Bayoumi, Waleed A. ; ElSayed, Magda A. ; Abouzeid, Laila A. ; Massoud, Mohammed A. M.

Chemical biology & drug design, 2022-07, Vol.100 (1), p.121-135 [Periódico revisado por pares]

England

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