1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors
Maurício Temotheo Tavares Arne Krüger; Sun Liu Rei Yan; Karoline de Barros Waitman; Vinícius de Morais Gomes; Daffiny Sumam de Oliveira; Franciarli Paz; Sebastian Hilscher; Mike Schutkowski; Wolfgang Sippl; Claudia Ruiz; Mônica Franco Zannini Junqueira Toledo; Antti Poso; Michael D Cameron; Thomas D Bannister; Thales Kronenberger; Roberto Parise Filho; Neuza Mariko Aymoto Hassimotto; João Agostinho Machado Neto; Giuseppe Palmisano; Carsten Wrenger
Scientific Reports London v. 13, n. 1, art. 21006, 20 p., 2023
London Nature Publishing Group 2023
Item não circula. Consulte sua biblioteca.(Acessar)
High target homology does not guarantee inhibition aminothiazoles emerge as inhibitors of Plasmodium falciparum
Sandra Johannsen Robin Matthias Gierse; Arne Kruger; Rachel L Edwards; Vittoria Nanna; Anna Fontana; Di Zhu; Tiziana Masini; Lais Pessanha de Carvalho; Mael Poizat Bart Kieftenbelt; Dana M Hodge Sophie Alvarez; Daan Bunt Antoine Lacour; Atanaz Shams; Kamila Anna Meissner; Edmarcia Elisa de Souza; Melloney Dröge; Bernard van Vilet Jack den Hartog Michael C. Hutter; Jana Held; Audrey R. Odom John Anna K. H. Hirsch; Carsten Wrenger
ACS Infectious Diseases Washington, DC v. 10, n. 3, p. 1000-1022, 2024
Washington, DC American Chemical Society 2024
Item não circula. Consulte sua biblioteca.(Acessar)