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Material Type: Artigo
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C–H activation reactions as useful tools for medicinal chemistsCaro-Diaz, Eduardo J.E. ; Urbano, Mariangela ; Buzard, Daniel J. ; Jones, Robert M.Bioorganic & medicinal chemistry letters, 2016-11, Vol.26 (22), p.5378-5383 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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A new target for Alzheimer’s disease: A small molecule SERCA activator is neuroprotective in vitro and improves memory and cognition in APP/PS1 miceKrajnak, Katherine ; Dahl, RussellBioorganic & medicinal chemistry letters, 2018-05, Vol.28 (9), p.1591-1594 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Design, synthesis and in vitro antimalarial activity of an acylhydrazone libraryMelnyk, Patricia ; Leroux, Virginie ; Sergheraert, Christian ; Grellier, PhilippeBioorganic & medicinal chemistry letters, 2006, Vol.16 (1), p.31-35 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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An antibacterial ortho-quinone diterpenoid and its derivatives from Caryopteris mongolicaSaruul, Erdenebileg ; Murata, Toshihiro ; Selenge, Erdenechimeg ; Sasaki, Kenroh ; Yoshizaki, Fumihiko ; Batkhuu, JavzanBioorganic & medicinal chemistry letters, 2015-06, Vol.25 (12), p.2555-2558 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Structure-based design of novel human Pin1 inhibitors (III): Optimizing affinity beyond the phosphate recognition pocketGuo, Chuangxing ; Hou, Xinjun ; Dong, Liming ; Marakovits, Joseph ; Greasley, Samantha ; Dagostino, Eleanor ; Ferre, RoseAnn ; Catherine Johnson, M. ; Humphries, Paul S. ; Li, Haitao ; Paderes, Genevieve D. ; Piraino, Joseph ; Kraynov, Eugenia ; Murray, Brion W.Bioorganic & medicinal chemistry letters, 2014-09, Vol.24 (17), p.4187-4191 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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New antioxidant polyphenols from the medicinal mushroom Inonotus obliquusLee, In-Kyoung ; Kim, Young-Sook ; Jang, Yoon-Woo ; Jung, Jin-Young ; Yun, Bong-SikBioorganic & medicinal chemistry letters, 2007-12, Vol.17 (24), p.6678-6681 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and antitumor activity of benzils related to combretastatin A-4Mousset, Céline ; Giraud, Anne ; Provot, Olivier ; Hamze, Abdallah ; Bignon, Jérôme ; Liu, Jian-Miao ; Thoret, Sylviane ; Dubois, Joëlle ; Brion, Jean-Daniel ; Alami, MouâdBioorganic & medicinal chemistry letters, 2008-06, Vol.18 (11), p.3266-3271 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Pterocarpans and flavanones from Sophora flavescens displaying potent neuraminidase inhibitionRyu, Young Bae ; Curtis-Long, Marcus J ; Kim, Jin Hyo ; Jeong, Seong Hun ; Yang, Min Suk ; Lee, Keun Woo ; Lee, Woo Song ; Park, Ki HunBioorganic & medicinal chemistry, 2008-12, Vol.18 (23), p.6046-6049 [Periódico revisado por pares]Amsterdam: ElsevierTexto completo disponível |
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Material Type: Artigo
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Triazole oxytocin antagonists: Identification of an aryloxyazetidine replacement for a biaryl substituentBrown, Alan ; Brown, T. Bruce ; Calabrese, Andrew ; Ellis, Dave ; Puhalo, Nicholas ; Ralph, Michael ; Watson, LesaBioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.516-520 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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The SARS-CoV-2 main protease as drug targetUllrich, Sven ; Nitsche, ChristophBioorganic & medicinal chemistry letters, 2020-09, Vol.30 (17), p.127377-127377, Article 127377 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |