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Material Type: Artigo
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Antimalarial activity of compounds comprising a primary benzene sulfonamide fragmentAndrews, Katherine T. ; Fisher, Gillian M. ; Sumanadasa, Subathdrage D.M. ; Skinner-Adams, Tina ; Moeker, Janina ; Lopez, Marie ; Poulsen, Sally-AnnBioorganic & medicinal chemistry letters, 2013-11, Vol.23 (22), p.6114-6117 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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In vitro inhibition of translation initiation by N,N′-diarylureas—potential anti-cancer agentsDenoyelle, Séverine ; Chen, Ting ; Chen, Limo ; Wang, Yibo ; Klosi, Edvin ; Halperin, José A. ; Aktas, Bertal H. ; Chorev, MichaelBioorganic & medicinal chemistry letters, 2012-01, Vol.22 (1), p.402-409 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Novel in vivo active anti-malarials based on a hydroxy-ethyl-amine scaffoldCiana, Claire-Lise ; Siegrist, Romain ; Aissaoui, Hamed ; Marx, Léo ; Racine, Sophie ; Meyer, Solange ; Binkert, Christoph ; de Kanter, Ruben ; Fischli, Christoph ; Wittlin, Sergio ; Boss, ChristophBioorganic & medicinal chemistry letters, 2013-02, Vol.23 (3), p.658-662 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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4-Thiophenoxy-2-trichloromethyquinazolines display in vitro selective antiplasmodial activity against the human malaria parasite Plasmodium falciparumVerhaeghe, Pierre ; Dumètre, Aurélien ; Castera-Ducros, Caroline ; Hutter, Sébastien ; Laget, Michèle ; Fersing, Cyril ; Prieri, Marion ; Yzombard, Julien ; Sifredi, France ; Rault, Sylvain ; Rathelot, Pascal ; Vanelle, Patrice ; Azas, NadineBioorganic & medicinal chemistry letters, 2011-10, Vol.21 (19), p.6003-6006 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Repurposing strategies for tropical disease drug discoveryKlug, Dana M. ; Gelb, Michael H. ; Pollastri, Michael P.Bioorganic & medicinal chemistry letters, 2016-06, Vol.26 (11), p.2569-2576 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compoundsÖztürk Sarikaya, Sevim Beyza ; Topal, Fevzi ; Şentürk, Murat ; Gülçin, İlhami ; Supuran, Claudiu T.Bioorganic & medicinal chemistry letters, 2011-07, Vol.21 (14), p.4259-4262 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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New pentasubstituted pyrrole hybrid atorvastatin–quinoline derivatives with antiplasmodial activityCarvalho, Rita C.C. ; Martins, Wagner A. ; Silva, Tayara P. ; Kaiser, Carlos R. ; Bastos, Mônica M. ; Pinheiro, Luiz C.S. ; Krettli, Antoniana U. ; Boechat, NúbiaBioorganic & medicinal chemistry letters, 2016-04, Vol.26 (8), p.1881-1884 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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1H-1,2,3-Triazole-tethered isatin-7-chloroquinoline and 3-hydroxy-indole-7-chloroquinoline conjugates: Synthesis and antimalarial evaluationRaj, Raghu ; Gut, Jiri ; Rosenthal, Philip J. ; Kumar, VipanBioorganic & medicinal chemistry letters, 2014-02, Vol.24 (3), p.756-759 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis, antimalarial and antitubercular activity of acetylenic chalconesHans, Renate H. ; Guantai, Eric M. ; Lategan, Carmen ; Smith, Peter J. ; Wan, Baojie ; Franzblau, Scott G. ; Gut, Jiri ; Rosenthal, Philip J. ; Chibale, KellyBioorganic & medicinal chemistry letters, 2010-02, Vol.20 (3), p.942-944 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and in vitro evaluation of hydrazinyl phthalazines against malaria parasite, Plasmodium falciparumSubramanian, Gowtham ; Babu Rajeev, C.P. ; Mohan, Chakrabhavi Dhananjaya ; Sinha, Ameya ; Chu, Trang T.T. ; Anusha, Sebastian ; Ximei, Huang ; Fuchs, Julian E. ; Bender, Andreas ; Rangappa, Kanchugarakoppal S. ; Chandramohanadas, Rajesh ; BasappaBioorganic & medicinal chemistry letters, 2016-07, Vol.26 (14), p.3300-3306 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |