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1
Phytogenic Polyphenols as Glycogen Phosphorylase Inhibitors: The Potential of Triterpenes and Flavonoids for Glycaemic Control in Type 2 Diabetes
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Phytogenic Polyphenols as Glycogen Phosphorylase Inhibitors: The Potential of Triterpenes and Flavonoids for Glycaemic Control in Type 2 Diabetes

Leonidas, Demetres D ; Hayes, Joseph M ; Kato, Atsushi ; Skamnaki, Vassiliki T ; Chatzileontiadou, Demetra S M ; Kantsadi, Anastassia L ; Kyriakis, Efthimios ; Chetter, Ben A ; Stravodimos, George A

Current medicinal chemistry, 2017-02, Vol.24 (4), p.384-403 [Periódico revisado por pares]

United Arab Emirates: Bentham Science Publishers Ltd

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2
Nicotinic cholinergic system and COVID-19: In silico evaluation of nicotinic acetylcholine receptor agonists as potential therapeutic interventions
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Artigo
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Nicotinic cholinergic system and COVID-19: In silico evaluation of nicotinic acetylcholine receptor agonists as potential therapeutic interventions

Alexandris, Nikolaos ; Lagoumintzis, George ; Chasapis, Christos T. ; Leonidas, Demetres D. ; Papadopoulos, Georgios E. ; Tzartos, Socrates J. ; Tsatsakis, Aristidis ; Eliopoulos, Elias ; Poulas, Konstantinos ; Farsalinos, Konstantinos

Toxicology reports, 2021-01, Vol.8, p.73-83 [Periódico revisado por pares]

Ireland: Elsevier B.V

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3
Naturally Occurring Pentacyclic Triterpenes as Inhibitors of Glycogen Phosphorylase: Synthesis, Structure−Activity Relationships, and X-ray Crystallographic Studies
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Naturally Occurring Pentacyclic Triterpenes as Inhibitors of Glycogen Phosphorylase: Synthesis, Structure−Activity Relationships, and X-ray Crystallographic Studies

Wen, Xiaoan ; Sun, Hongbin ; Liu, Jun ; Cheng, Keguang ; Zhang, Pu ; Zhang, Liying ; Hao, Jia ; Zhang, Luyong ; Ni, Peizhou ; Zographos, Spyros E ; Leonidas, Demetres D ; Alexacou, Kyra-Melinda ; Gimisis, Thanasis ; Hayes, Joseph M ; Oikonomakos, Nikos G

Journal of medicinal chemistry, 2008-06, Vol.51 (12), p.3540-3554 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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4
High Consistency of Structure-Based Design and X-Ray Crystallography: Design, Synthesis, Kinetic Evaluation and Crystallographic Binding Mode Determination of Biphenyl- N -acyl-β-d-Glucopyranosylamines as Glycogen Phosphorylase Inhibitors
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High Consistency of Structure-Based Design and X-Ray Crystallography: Design, Synthesis, Kinetic Evaluation and Crystallographic Binding Mode Determination of Biphenyl- N -acyl-β-d-Glucopyranosylamines as Glycogen Phosphorylase Inhibitors

Fischer, Thomas ; Koulas, Symeon M ; Tsagkarakou, Anastasia S ; Kyriakis, Efthimios ; Stravodimos, George A ; Skamnaki, Vassiliki T ; Liggri, Panagiota G V ; Zographos, Spyros E ; Riedl, Rainer ; Leonidas, Demetres D

Molecules (Basel, Switzerland), 2019-04, Vol.24 (7), p.1322 [Periódico revisado por pares]

Switzerland: MDPI AG

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5
Computation as a Tool for Glycogen Phosphorylase Inhibitor Design
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Computation as a Tool for Glycogen Phosphorylase Inhibitor Design

Hayes, Joseph M ; Leonidas, Demetres D

Mini reviews in medicinal chemistry, 2010-10, Vol.10 (12), p.1156-1174 [Periódico revisado por pares]

Netherlands: Bentham Science Publishers Ltd

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6
Biochemical and in silico identification of the active site and the catalytic mechanism of the circadian deadenylase HESPERIN
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Artigo
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Biochemical and in silico identification of the active site and the catalytic mechanism of the circadian deadenylase HESPERIN

Beta, Rafailia A. A. ; Kyritsis, Athanasios ; Douka, Veroniki ; Papanastasi, Eirini ; Rizouli, Marianna ; Leonidas, Demetres D. ; Vlachakis, Dimitrios ; Balatsos, Nikolaos A. A.

FEBS open bio, 2022-05, Vol.12 (5), p.1036-1049 [Periódico revisado por pares]

England: John Wiley & Sons, Inc

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7
Oxidation of human serum albumin exhibits inter-individual variability after an ultra-marathon mountain race
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Oxidation of human serum albumin exhibits inter-individual variability after an ultra-marathon mountain race

Spanidis, Ypatios ; Priftis, Alexandros ; Stagos, Dimitrios ; Stravodimos, George A ; Leonidas, Demetres D ; Spandidos, Demetrios A ; Tsatsakis, Aristides M ; Kouretas, Demetrios

Experimental and therapeutic medicine, 2017-05, Vol.13 (5), p.2382-2390

Greece: Spandidos Publications

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8
Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitors
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Artigo
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Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitors

Benltifa, Mahmoud ; Hayes, Joseph M. ; Vidal, Sébastien ; Gueyrard, David ; Goekjian, Peter G. ; Praly, Jean-Pierre ; Kizilis, Gregory ; Tiraidis, Costas ; Alexacou, Kyra-Melinda ; Chrysina, Evangelia D. ; Zographos, Spyros E. ; Leonidas, Demetres D. ; Archontis, Georgios ; Oikonomakos, Nikos G.

Bioorganic & medicinal chemistry, 2009-10, Vol.17 (20), p.7368-7380 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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9
Affinity Crystallography Reveals the Bioactive Compounds of Industrial Juicing Byproducts of Punica granatum for Glycogen Phosphorylase
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Artigo
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Affinity Crystallography Reveals the Bioactive Compounds of Industrial Juicing Byproducts of Punica granatum for Glycogen Phosphorylase

Stravodimos, George A ; Kantsadi, Anastassia L ; Apostolou, Anna ; Kyriakis, Efthimios ; Kafaski-Kanelli, Vassiliki-Nafsika ; Solovou, Theodora ; Gatzona, Pagona ; Liggri, Panagiota G V ; Theofanous, Stavroula ; Gorgogietas, Vyron A ; Kissa, Apostolia ; Psachoula, Chariklia ; Lemonakis, Angelos ; Chatzileontiadou, Demetra S M ; Psarra, Anna-Maria G ; Skamnaki, Vassiliki T ; Haroutounian, Serkos A ; Leonidas, Demetres D

Current drug discovery technologies, 2018, Vol.15 (1), p.41-53 [Periódico revisado por pares]

United Arab Emirates: Bentham Science Publishers Ltd

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10
Molecular Cloning, Carbohydrate Specificity and the Crystal Structure of Two Sclerotium rolfsii Lectin Variants
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Artigo
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Molecular Cloning, Carbohydrate Specificity and the Crystal Structure of Two Sclerotium rolfsii Lectin Variants

Peppa, Vassiliki I ; Venkat, Hemalatha ; Kantsadi, Anastassia L ; Inamdar, Shashikala R ; Bhat, Ganapati G ; Eligar, Sachin ; Shivanand, Anupama ; Chachadi, Vishwanath B ; Satisha, Gonchigar J ; Swamy, Bale M ; Skamnaki, Vassiliki T ; Zographos, Spyridon E ; Leonidas, Demetres D

Molecules (Basel, Switzerland), 2015-06, Vol.20 (6), p.10848-10865 [Periódico revisado por pares]

Switzerland: MDPI AG

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