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Refinado por: Nome da Publicação: Bioorganic & Medicinal Chemistry remover
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11
Development of matrix metalloproteinase-13 inhibitors – A structure-activity/structure-property relationship study
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Development of matrix metalloproteinase-13 inhibitors – A structure-activity/structure-property relationship study

Fuerst, Rita ; Yong Choi, Jun ; Knapinska, Anna M. ; Smith, Lyndsay ; Cameron, Michael D. ; Ruiz, Claudia ; Fields, Gregg B. ; Roush, William R.

Bioorganic & medicinal chemistry, 2018-10, Vol.26 (18), p.4984-4995 [Periódico revisado por pares]

England: Elsevier Ltd

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12
Potent anti-melanogenic activity and favorable toxicity profile of selected 4-phenyl hydroxycoumarins in the zebrafish model and the computational molecular modeling studies
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Artigo
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Potent anti-melanogenic activity and favorable toxicity profile of selected 4-phenyl hydroxycoumarins in the zebrafish model and the computational molecular modeling studies

Veselinović, Jovana B. ; Veselinović, Aleksandar M. ; Ilic-Tomic, Tatjana ; Davis, Reeta ; O'Connor, Kevin ; Pavic, Aleksandar ; Nikodinovic-Runic, Jasmina

Bioorganic & medicinal chemistry, 2017-12, Vol.25 (24), p.6286-6296 [Periódico revisado por pares]

England: Elsevier Ltd

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13
Using in vitro ADME data for lead compound selection: An emphasis on PAMPA pH 5 permeability and oral bioavailability
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Using in vitro ADME data for lead compound selection: An emphasis on PAMPA pH 5 permeability and oral bioavailability

Williams, Jordan ; Siramshetty, Vishal ; Nguyễn, Ðắc-Trung ; Padilha, Elias Carvalho ; Kabir, Md ; Yu, Kyeong-Ri ; Wang, Amy Q. ; Zhao, Tongan ; Itkin, Misha ; Shinn, Paul ; Mathé, Ewy A. ; Xu, Xin ; Shah, Pranav

Bioorganic & medicinal chemistry, 2022-02, Vol.56, p.116588-116588, Article 116588 [Periódico revisado por pares]

England: Elsevier Ltd

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14
Synthesis and biological activity of thieno[3,2-d]pyrimidines as potent JAK3 inhibitors for the treatment of idiopathic pulmonary fibrosis
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Artigo
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Synthesis and biological activity of thieno[3,2-d]pyrimidines as potent JAK3 inhibitors for the treatment of idiopathic pulmonary fibrosis

Zhu, Yanming ; Zheng, Xu ; Wang, Changyuan ; Sun, Xiuli ; Sun, Huijun ; Ma, Tengyue ; Li, Yanxia ; Liu, Kexin ; Chen, Lixue ; Ma, Xiaodong

Bioorganic & medicinal chemistry, 2020-01, Vol.28 (2), p.115254, Article 115254 [Periódico revisado por pares]

England: Elsevier Ltd

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15
Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies
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Artigo
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Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies

Sarigol, Deniz ; Uzgoren-Baran, Ayse ; Tel, Banu Cahide ; Somuncuoglu, Elif Inci ; Kazkayasi, Inci ; Ozadali-Sari, Keriman ; Unsal-Tan, Oya ; Okay, Gurol ; Ertan, Mevlut ; Tozkoparan, Birsen

Bioorganic & medicinal chemistry, 2015-05, Vol.23 (10), p.2518-2528 [Periódico revisado por pares]

England: Elsevier Ltd

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16
Cannabidiol (CBD) and its analogs: a review of their effects on inflammation
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Cannabidiol (CBD) and its analogs: a review of their effects on inflammation

Burstein, Sumner

Bioorganic & medicinal chemistry, 2015-04, Vol.23 (7), p.1377-1385 [Periódico revisado por pares]

England: Elsevier Ltd

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17
Synthesis, in vitro and in vivo biological evaluation of novel graveolinine derivatives as potential anti-Alzheimer agents
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Artigo
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Synthesis, in vitro and in vivo biological evaluation of novel graveolinine derivatives as potential anti-Alzheimer agents

Luo, Wen ; Lv, Jian-Wu ; Wang, Ting ; Zhang, Zhi-Yang ; Guo, Hui-Yan ; Song, Zhi-Yi ; Wang, Chao-Jie ; Ma, Jing ; Chen, Yi-ping

Bioorganic & medicinal chemistry, 2020-01, Vol.28 (1), p.115190, Article 115190 [Periódico revisado por pares]

England: Elsevier Ltd

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18
Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine
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Artigo
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Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine

da Silva, Vinícius Barros Ribeiro ; Campos, Bruna Rafaella Koresch Leiva ; de Oliveira, Jamerson Ferreira ; Decout, Jean-Luc ; do Carmo Alves de Lima, Maria

Bioorganic & medicinal chemistry, 2017-07, Vol.25 (13), p.3259-3277 [Periódico revisado por pares]

England: Elsevier Ltd

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19
Discovery of pyrrolo[3,2-c]quinoline-4-one derivatives as novel hedgehog signaling inhibitors
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Artigo
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Discovery of pyrrolo[3,2-c]quinoline-4-one derivatives as novel hedgehog signaling inhibitors

Ohashi, Tomohiro ; Oguro, Yuya ; Tanaka, Toshio ; Shiokawa, Zenyu ; Shibata, Sachio ; Sato, Yoshihiko ; Yamakawa, Hiroko ; Hattori, Harumi ; Yamamoto, Yukiko ; Kondo, Shigeru ; Miyamoto, Maki ; Tojo, Hideaki ; Baba, Atsuo ; Sasaki, Satoshi

Bioorganic & medicinal chemistry, 2012-09, Vol.20 (18), p.5496-5506 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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20
Discovery of novel N-(5-(arylcarbonyl)thiazol-2-yl)amides and N-(5-(arylcarbonyl)thiophen-2-yl)amides as potent RORγt inhibitors
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Artigo
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Discovery of novel N-(5-(arylcarbonyl)thiazol-2-yl)amides and N-(5-(arylcarbonyl)thiophen-2-yl)amides as potent RORγt inhibitors

Wang, Yonghui ; Cai, Wei ; Zhang, Guifeng ; Yang, Ting ; Liu, Qian ; Cheng, Yaobang ; Zhou, Ling ; Ma, Yingli ; Cheng, Ziqiang ; Lu, Sijie ; Zhao, Yong-Gang ; Zhang, Wei ; Xiang, Zhijun ; Wang, Shuai ; Yang, Liuqing ; Wu, Qianqian ; Orband-Miller, Lisa A. ; Xu, Yan ; Zhang, Jing ; Gao, Ruina ; Huxdorf, Melanie ; Xiang, Jia-Ning ; Zhong, Zhong ; Elliott, John D. ; Leung, Stewart ; Lin, Xichen

Bioorganic & medicinal chemistry, 2014-01, Vol.22 (2), p.692-702 [Periódico revisado por pares]

England: Elsevier Ltd

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