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Refinado por: Nome da Publicação: Bioorganic & Medicinal Chemistry remover
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21
Discovery of novel N-(5-(arylcarbonyl)thiazol-2-yl)amides and N-(5-(arylcarbonyl)thiophen-2-yl)amides as potent RORγt inhibitors
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Discovery of novel N-(5-(arylcarbonyl)thiazol-2-yl)amides and N-(5-(arylcarbonyl)thiophen-2-yl)amides as potent RORγt inhibitors

Wang, Yonghui ; Cai, Wei ; Zhang, Guifeng ; Yang, Ting ; Liu, Qian ; Cheng, Yaobang ; Zhou, Ling ; Ma, Yingli ; Cheng, Ziqiang ; Lu, Sijie ; Zhao, Yong-Gang ; Zhang, Wei ; Xiang, Zhijun ; Wang, Shuai ; Yang, Liuqing ; Wu, Qianqian ; Orband-Miller, Lisa A. ; Xu, Yan ; Zhang, Jing ; Gao, Ruina ; Huxdorf, Melanie ; Xiang, Jia-Ning ; Zhong, Zhong ; Elliott, John D. ; Leung, Stewart ; Lin, Xichen

Bioorganic & medicinal chemistry, 2014-01, Vol.22 (2), p.692-702 [Periódico revisado por pares]

England: Elsevier Ltd

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22
Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation
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Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation

Papadopoulou, Maria V. ; Bloomer, William D. ; Rosenzweig, Howard S. ; O’Shea, Ivan P. ; Wilkinson, Shane R. ; Kaiser, Marcel ; Chatelain, Eric ; Ioset, Jean-Robert

Bioorganic & medicinal chemistry, 2015-10, Vol.23 (19), p.6467-6476 [Periódico revisado por pares]

England: Elsevier Ltd

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23
Structure-based design, synthesis, and biological evaluation of imidazo[1,2-b]pyridazine-based p38 MAP kinase inhibitors
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Artigo
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Structure-based design, synthesis, and biological evaluation of imidazo[1,2-b]pyridazine-based p38 MAP kinase inhibitors

Kaieda, Akira ; Takahashi, Masashi ; Takai, Takafumi ; Goto, Masayuki ; Miyazaki, Takahiro ; Hori, Yuri ; Unno, Satoko ; Kawamoto, Tomohiro ; Tanaka, Toshimasa ; Itono, Sachiko ; Takagi, Terufumi ; Hamada, Teruki ; Shirasaki, Mikio ; Okada, Kengo ; Snell, Gyorgy ; Bragstad, Ken ; Sang, Bi-Ching ; Uchikawa, Osamu ; Miwatashi, Seiji

Bioorganic & medicinal chemistry, 2018-02, Vol.26 (3), p.647-660 [Periódico revisado por pares]

England: Elsevier Ltd

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24
Synthesis and antifungal activity of substituted salicylaldehyde hydrazones, hydrazides and sulfohydrazides
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Synthesis and antifungal activity of substituted salicylaldehyde hydrazones, hydrazides and sulfohydrazides

Backes, Gregory L. ; Neumann, Donna M. ; Jursic, Branko S.

Bioorganic & medicinal chemistry, 2014-09, Vol.22 (17), p.4629-4636 [Periódico revisado por pares]

England: Elsevier Ltd

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25
Design, synthesis and anticonvulsant properties of new N-Mannich bases derived from 3-phenylpyrrolidine-2,5-diones
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Design, synthesis and anticonvulsant properties of new N-Mannich bases derived from 3-phenylpyrrolidine-2,5-diones

Kamiński, Krzysztof ; Obniska, Jolanta ; Chlebek, Iwona ; Wiklik, Beata ; Rzepka, Sabina

Bioorganic & medicinal chemistry, 2013-11, Vol.21 (21), p.6821-6830 [Periódico revisado por pares]

England: Elsevier Ltd

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26
Biphenyloxy-alkyl-piperidine and azepane derivatives as histamine H 3 receptor ligands
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Biphenyloxy-alkyl-piperidine and azepane derivatives as histamine H 3 receptor ligands

Łażewska, Dorota ; Kaleta, Maria ; Schwed, J Stephan ; Karcz, Tadeusz ; Mogilski, Szczepan ; Latacz, Gniewomir ; Olejarz, Agnieszka ; Siwek, Agata ; Kubacka, Monika ; Lubelska, Annamaria ; Honkisz, Ewelina ; Handzlik, Jadwiga ; Filipek, Barbara ; Stark, Holger ; Kieć-Kononowicz, Katarzyna

Bioorganic & medicinal chemistry, 2017-10, Vol.25 (20), p.5341 [Periódico revisado por pares]

England

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27
Nanoparticle-macrophage interactions: A balance between clearance and cell-specific targeting
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Nanoparticle-macrophage interactions: A balance between clearance and cell-specific targeting

Rattan, Rahul ; Bhattacharjee, Somnath ; Zong, Hong ; Swain, Corban ; Siddiqui, Muneeb A. ; Visovatti, Scott H. ; Kanthi, Yogendra ; Desai, Sajani ; Pinsky, David J. ; Goonewardena, Sascha N.

Bioorganic & medicinal chemistry, 2017-08, Vol.25 (16), p.4487-4496 [Periódico revisado por pares]

England: Elsevier Ltd

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28
Design, synthesis and biological evaluation of novel carbamates as potential inhibitors of acetylcholinesterase and butyrylcholinesterase
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Design, synthesis and biological evaluation of novel carbamates as potential inhibitors of acetylcholinesterase and butyrylcholinesterase

Wu, Jie ; Pistolozzi, Marco ; Liu, Siyu ; Tan, Wen

Bioorganic & medicinal chemistry, 2020-03, Vol.28 (5), p.115324, Article 115324 [Periódico revisado por pares]

England

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29
Design, synthesis, and antitumor activity evaluation of novel acyl sulfonamide spirodienones
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Design, synthesis, and antitumor activity evaluation of novel acyl sulfonamide spirodienones

Chen, Chen ; Luo, Yang ; Yin, Honglu ; Zhong, Qiu ; Zheng, Shilong ; Liu, Rui ; Zhao, Chong ; Wang, Guangdi ; He, Ling

Bioorganic & medicinal chemistry, 2022-04, Vol.60, p.116626-116626, Article 116626 [Periódico revisado por pares]

England: Elsevier Ltd

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30
Structure–activity relationship of flavonoids as influenza virus neuraminidase inhibitors and their in vitro anti-viral activities
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Structure–activity relationship of flavonoids as influenza virus neuraminidase inhibitors and their in vitro anti-viral activities

Liu, Ai-Lin ; Wang, Hai-Di ; Lee, Simon MingYuen ; Wang, Yi-Tao ; Du, Guan-Hua

Bioorganic & medicinal chemistry, 2008-08, Vol.16 (15), p.7141-7147 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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