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1
Synthesis and antidiabetic activity of 2,5-disubstituted-3-imidazol-2-yl-pyrrolo[2,3- b]pyridines and thieno[2,3- b]pyridines
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Synthesis and antidiabetic activity of 2,5-disubstituted-3-imidazol-2-yl-pyrrolo[2,3- b]pyridines and thieno[2,3- b]pyridines

Bahekar, Rajesh H. ; Jain, Mukul R. ; Jadav, Pradip A. ; Prajapati, Vijay M. ; Patel, Dipam N. ; Gupta, Arun A. ; Sharma, Ajay ; Tom, Robby ; Bandyopadhya, Debdutta ; Modi, Honey ; Patel, Pankaj R.

Bioorganic & medicinal chemistry, 2007-11, Vol.15 (21), p.6782-6795 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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2
Discovery of novel analgesic and anti-inflammatory 3-arylamine-imidazo[1,2- a]pyridine symbiotic prototypes
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Discovery of novel analgesic and anti-inflammatory 3-arylamine-imidazo[1,2- a]pyridine symbiotic prototypes

Lacerda, Renata B. ; de Lima, Cleverton K.F. ; da Silva, Leandro L. ; Romeiro, Nelilma C. ; Miranda, Ana Luisa P. ; Barreiro, Eliezer J. ; Fraga, Carlos A.M.

Bioorganic & medicinal chemistry, 2009, Vol.17 (1), p.74-84 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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3
Synthesis and pharmacological evaluation of thieno[2,3- b]pyridine derivatives as novel c-Src inhibitors
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Synthesis and pharmacological evaluation of thieno[2,3- b]pyridine derivatives as novel c-Src inhibitors

Pevet, Isabelle ; Brulé, Cédric ; Tizot, André ; Gohier, Arnaud ; Cruzalegui, Francisco ; Boutin, Jean A. ; Goldstein, Solo

Bioorganic & medicinal chemistry, 2011-04, Vol.19 (8), p.2517-2528 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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4
Design, synthesis, and biological evaluation of substituted- N-(thieno[2,3- b]pyridin-3-yl)-guanidines, N-(1 H-pyrrolo[2,3- b]pyridin-3-yl)-guanidines, and N-(1 H-indol-3-yl)-guanidines
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Design, synthesis, and biological evaluation of substituted- N-(thieno[2,3- b]pyridin-3-yl)-guanidines, N-(1 H-pyrrolo[2,3- b]pyridin-3-yl)-guanidines, and N-(1 H-indol-3-yl)-guanidines

Bahekar, Rajesh H. ; Jain, Mukul R. ; Goel, Ashish ; Patel, Dipam N. ; Prajapati, Vijay M. ; Gupta, Arun A. ; Jadav, Pradip A. ; Patel, Pankaj R.

Bioorganic & medicinal chemistry, 2007-05, Vol.15 (9), p.3248-3265 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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5
Synthesis and antiproliferative activity of pyrrolo[3,2- b]pyridine derivatives against melanoma
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Synthesis and antiproliferative activity of pyrrolo[3,2- b]pyridine derivatives against melanoma

Kim, Hee Jin ; Jung, Myung-Ho ; Kim, Hwan ; El-Gamal, Mohammed I. ; Sim, Tae Bo ; Lee, So Ha ; Hong, Jun Hee ; Hah, Jung-Mi ; Cho, Jung-Hyuck ; Choi, Jung Hoon ; Yoo, Kyung Ho ; Oh, Chang-Hyun

Bioorganic & medicinal chemistry letters, 2010, Vol.20 (1), p.413-417 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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6
Synthesis of 3-(1 H-benzimidazol-2-yl)-5-isoquinolin-4-ylpyrazolo[1,2- b]pyridine, a potent cyclin dependent kinase 1 (CDK1) inhibitor
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Synthesis of 3-(1 H-benzimidazol-2-yl)-5-isoquinolin-4-ylpyrazolo[1,2- b]pyridine, a potent cyclin dependent kinase 1 (CDK1) inhibitor

Huang, Shenlin ; Lin, Ronghui ; Yu, Yang ; Lu, Yanhua ; Connolly, Peter J. ; Chiu, George ; Li, Shengjian ; Emanuel, Stuart L. ; Middleton, Steven A.

Bioorganic & medicinal chemistry letters, 2007-03, Vol.17 (5), p.1243-1245 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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7
Inhibition of eEF2-K by thieno[2,3- b]pyridine analogues
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Inhibition of eEF2-K by thieno[2,3- b]pyridine analogues

Lockman, Jeffrey W. ; Reeder, Matthew D. ; Suzuki, Kazuyuki ; Ostanin, Kirill ; Hoff, Ryan ; Bhoite, Leena ; Austin, Harry ; Baichwal, Vijay ; Adam Willardsen, J.

Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (7), p.2283-2286 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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8
Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitors
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Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitors

Han, Sun-Young ; Choi, Jie Won ; Yang, Jeon ; Chae, Chong Hack ; Lee, Jongkook ; Jung, Heejung ; Lee, Kwangho ; Ha, Jae Du ; Kim, Hyoung Rae ; Cho, Sung Yun

Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (8), p.2837-2842 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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9
Positive Allosteric Modulation of mGluR5 Receptors Facilitates Extinction of a Cocaine Contextual Memory
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Positive Allosteric Modulation of mGluR5 Receptors Facilitates Extinction of a Cocaine Contextual Memory

Gass, Justin T ; Olive, M. Foster

Biological psychiatry (1969), 2009-04, Vol.65 (8), p.717-720 [Periódico revisado por pares]

New York, NY: Elsevier Inc

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10
Discovery of a novel and potent series of thieno[3,2- b]pyridine-based inhibitors of c-Met and VEGFR2 tyrosine kinases
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Discovery of a novel and potent series of thieno[3,2- b]pyridine-based inhibitors of c-Met and VEGFR2 tyrosine kinases

Claridge, Stephen ; Raeppel, Franck ; Granger, Marie-Claude ; Bernstein, Naomy ; Saavedra, Oscar ; Zhan, Lijie ; Llewellyn, David ; Wahhab, Amal ; Deziel, Robert ; Rahil, Jubrail ; Beaulieu, Normand ; Nguyen, Hannah ; Dupont, Isabelle ; Barsalou, Annie ; Beaulieu, Carole ; Chute, Ian ; Gravel, Serge ; Robert, Marie-France ; Lefebvre, Sylvain ; Dubay, Marja ; Pascal, Roussen ; Gillespie, Jeff ; Jin, Zhiyun ; Wang, James ; Besterman, Jeffrey M. ; MacLeod, A. Robert ; Vaisburg, Arkadii

Bioorganic & medicinal chemistry, 2008-05, Vol.18 (9), p.2793-2798 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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