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1
Urinary and biliary excretion of metabolites of halothane in dogs
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Artigo
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Urinary and biliary excretion of metabolites of halothane in dogs

SAKAI, T ; YOSHIDA, H ; FUKUI, A ; TAKAORI, M

Drug metabolism and disposition, 1991-03, Vol.19 (2), p.419-422 [Periódico revisado por pares]

Bethesda, MD: American Society for Pharmacology and Experimental Therapeutics

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2
METABOLISM OF ENFLURANE IN DOGS
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Artigo
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METABOLISM OF ENFLURANE IN DOGS

SAKAI, T ; TAKAORI, M ; YOSHIDA, H

Drug metabolism and disposition, 1992-01, Vol.20 (1), p.127-129 [Periódico revisado por pares]

BETHESDA: Amer Soc Pharmacology Experimental Therapeutics

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3
Disposition of the novel anticancer agent vinorelbine ditartrate following intravenous administration in mice, rats and dogs
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Artigo
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Disposition of the novel anticancer agent vinorelbine ditartrate following intravenous administration in mice, rats and dogs

Kobayashi, S ; Sakai, T ; Dalrymple, P D ; Wood, S G ; Chasseaud, L F

Arzneimittel-Forschung, 1993-12, Vol.43 (12), p.1367

Germany

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4
Bronchodilating and cardiovascular effects of intraduodenally and orally administered clenbuterol in dogs
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Artigo
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Bronchodilating and cardiovascular effects of intraduodenally and orally administered clenbuterol in dogs

Kato, H ; Nakayama, K ; Takata, Y ; Kurihara, J ; Sakai, T ; Iwata, K ; Yamamoto, I

Arzneimittel-Forschung, 1985, Vol.35 (7), p.1037

Germany

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5
Species differences in vacuolation of the choroid plexus induced by the piperidine-ring drug disobutamide in the rat, dog, and monkey
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Artigo
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Species differences in vacuolation of the choroid plexus induced by the piperidine-ring drug disobutamide in the rat, dog, and monkey

Koizumi, Haruko ; Watanabe, Mitsutoshi ; Numata, Hiroaki ; Sakai, Tadashi ; Morishita, Hiroshi

Toxicology and applied pharmacology, 1986-06, Vol.84 (1), p.125-148 [Periódico revisado por pares]

San Diego, CA: Elsevier Inc

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6
Interspecies Differences in Pharmacokinetics of an Antiallergic Agent, 1-(2-Ethoxyethyl)-2-(hexahydro-4-methyl-1, 4-diazepin-1-yl)benzimidazole Difumarate (KG-2413) after Intravenous Administration to Rats, Guinea Pigs and Dogs
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Artigo
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Interspecies Differences in Pharmacokinetics of an Antiallergic Agent, 1-(2-Ethoxyethyl)-2-(hexahydro-4-methyl-1, 4-diazepin-1-yl)benzimidazole Difumarate (KG-2413) after Intravenous Administration to Rats, Guinea Pigs and Dogs

SAKAI, Takanori ; HAMADA, Tsukasa ; AWATA, Norio ; WATANABE, Jun

Chemical and Pharmaceutical Bulletin, 1989/03/25, Vol.37(3), pp.753-756 [Periódico revisado por pares]

Tokyo: The Pharmaceutical Society of Japan

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7
Pharmacokinetics of an Antiallergic Agent, 1-(2-Ethoxyethyl)-2-(hexahydro-4-methyl-1H-1, 4-diazepin-1-yl)-1H-benzimidazole Difumarate (KG-2413) after Oral Administration : Interspecies Differences in Rats, Guinea Pigs and Dogs
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Artigo
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Pharmacokinetics of an Antiallergic Agent, 1-(2-Ethoxyethyl)-2-(hexahydro-4-methyl-1H-1, 4-diazepin-1-yl)-1H-benzimidazole Difumarate (KG-2413) after Oral Administration : Interspecies Differences in Rats, Guinea Pigs and Dogs

SAKAI, Takanori ; HAMADA, Tsukasa ; AWATA, Norio ; WATANABE, Jun

Journal of Pharmacobio-Dynamics, 1989, Vol.12(9), pp.530-536

Tokyo: The Pharmaceutical Society of Japan

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8
Structure−Activity Relationship Study and Drug Profile of N-(4-Fluorophenylsulfonyl)-l-valyl-l-leucinal (SJA6017) as a Potent Calpain Inhibitor
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Artigo
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Structure−Activity Relationship Study and Drug Profile of N-(4-Fluorophenylsulfonyl)-l-valyl-l-leucinal (SJA6017) as a Potent Calpain Inhibitor

Inoue, Jun ; Nakamura, Masayuki ; Cui, Ying-She ; Sakai, Yusuke ; Sakai, Osamu ; Hill, Jeanette R ; Wang, Kevin K. W ; Yuen, Po-Wai

Journal of medicinal chemistry, 2003-02, Vol.46 (5), p.868-871 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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9
Impact of Intestinal Glucuronidation on the Pharmacokinetics of Raloxifene
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Artigo
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Impact of Intestinal Glucuronidation on the Pharmacokinetics of Raloxifene

KOSAKA, Keigo ; SAKAI, Norifumi ; KUME, Toshiyuki ; ENDO, Yuya ; FUKUHARA, Yuga ; TSUDA-TSUKIMOTO, Minoru ; OHTSUKA, Tatsuyuki ; KINO, Ichiro ; TANIMOTO, Tomohiko ; TAKEBA, Naomi ; TAKAHASHI, Masakatsu

Drug metabolism and disposition, 2011-09, Vol.39 (9), p.1495-1502 [Periódico revisado por pares]

Bethesda, MD: American Society for Pharmacology and Experimental Therapeutics

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10
2-({6-[(3R)-3-amino-3-methylpiperidine-1-yl]-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidine-5-yl}methyl)-4-fluorobenzonitrile (DSR-12727): A potent, orally active dipeptidyl peptidase IV inhibitor without mechanism-based inactivation of CYP3A
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Artigo
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2-({6-[(3R)-3-amino-3-methylpiperidine-1-yl]-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidine-5-yl}methyl)-4-fluorobenzonitrile (DSR-12727): A potent, orally active dipeptidyl peptidase IV inhibitor without mechanism-based inactivation of CYP3A

Nishio, Yukihiro ; Kimura, Hidenori ; Sawada, Naoyuki ; Sugaru, Eiji ; Horiguchi, Masakuni ; Ono, Michiko ; Furuta, Yudai ; Sakai, Mutsuko ; Masui, Yumi ; Otani, Misato ; Hashizuka, Takahiko ; Honda, Yayoi ; Deguchi, Jiro ; Nakagawa, Tsutomu ; Nakahira, Hiroyuki

Bioorganic & medicinal chemistry, 2011-09, Vol.19 (18), p.5490-5499 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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