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Material Type: Artigo
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Outcomes of Alzheimer's disease therapy with acetylcholinesterase inhibitors and memantineZemek, Filip ; Drtinova, Lucie ; Nepovimova, Eugenie ; Sepsova, Vendula ; Korabecny, Jan ; Klimes, Jiri ; Kuca, KamilExpert opinion on drug safety, 2014-06, Vol.13 (6), p.759-774 [Periódico revisado por pares]London: Informa UK, LtdSem texto completo |
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2 |
Material Type: Artigo
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Bis-Amiridines as Acetylcholinesterase and Butyrylcholinesterase Inhibitors: N -Functionalization Determines the Multitarget Anti-Alzheimer's Activity ProfileMakhaeva, Galina F ; Kovaleva, Nadezhda V ; Boltneva, Natalia P ; Rudakova, Elena V ; Lushchekina, Sofya V ; Astakhova, Tatiana Yu ; Serkov, Igor V ; Proshin, Alexey N ; Radchenko, Eugene V ; Palyulin, Vladimir A ; Korabecny, Jan ; Soukup, Ondrej ; Bachurin, Sergey O ; Richardson, Rudy JMolecules (Basel, Switzerland), 2022-02, Vol.27 (3), p.1060 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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3 |
Material Type: Artigo
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Oxime K074 - in vitro and in silico reactivation of acetylcholinesterase inhibited by nerve agents and pesticidesKuca, Kamil ; Musilek, Kamil ; Jun, Daniel ; Nepovimova, Eugenie ; Soukup, Ondrej ; Korabecny, Jan ; França, Tanos C. C. ; de Castro, Alexandre A. ; Krejcar, Ondrej ; da Cunha, Elaine F. F. ; Ramalho, Teodorico C.Toxin reviews, 2020-04, Vol.39 (2), p.157-166 [Periódico revisado por pares]Taylor & FrancisSem texto completo |
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4 |
Material Type: Artigo
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Development of versatile and potent monoquaternary reactivators of acetylcholinesteraseGorecki, Lukas ; Hepnarova, Vendula ; Karasova, Jana Zdarova ; Hrabinova, Martina ; Courageux, Charlotte ; Dias, José ; Kucera, Tomas ; Kobrlova, Tereza ; Muckova, Lubica ; Prchal, Lukas ; Malinak, David ; Jun, Daniel ; Musilek, Kamil ; Worek, Franz ; Nachon, Florian ; Soukup, Ondrej ; Korabecny, JanArchives of toxicology, 2021-03, Vol.95 (3), p.985-1001 [Periódico revisado por pares]Berlin/Heidelberg: Springer Berlin HeidelbergTexto completo disponível |
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5 |
Material Type: Artigo
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Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivatorsMalinak, David ; Dolezal, Rafael ; Hepnarova, Vendula ; Hozova, Miroslava ; Andrys, Rudolf ; Bzonek, Petr ; Racakova, Veronika ; Korabecny, Jan ; Gorecki, Lukas ; Mezeiova, Eva ; Psotka, Miroslav ; Jun, Daniel ; Kuca, Kamil ; Musilek, KamilJournal of enzyme inhibition and medicinal chemistry, 2020-01, Vol.35 (1), p.478-488 [Periódico revisado por pares]England: Taylor & FrancisTexto completo disponível |
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Material Type: Artigo
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Non-covalent acetylcholinesterase inhibitors: In vitro screening and molecular modeling for novel selective insecticidesHepnarova, Vendula ; Hrabinova, Martina ; Muckova, Lubica ; Kucera, Tomas ; Schmidt, Monika ; Dolezal, Rafael ; Gorecki, Lukas ; Hrabcova, Veronika ; Korabecny, Jan ; Mezeiova, Eva ; Jun, Daniel ; Pejchal, JaroslavToxicology in vitro, 2022-12, Vol.85, p.105463-105463, Article 105463 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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Progress in acetylcholinesterase reactivators and in the treatment of organophosphorus intoxication: a patent review (2006-2016)Gorecki, Lukas ; Korabecny, Jan ; Musilek, Kamil ; Nepovimova, Eugenie ; Malinak, David ; Kucera, Tomas ; Dolezal, Rafael ; Jun, Daniel ; Soukup, Ondrej ; Kuca, KamilExpert opinion on therapeutic patents, 2017-09, Vol.27 (9), p.971-985 [Periódico revisado por pares]England: Taylor & FrancisSem texto completo |
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8 |
Material Type: Artigo
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From Pyridinium-based to Centrally Active Acetylcholinesterase ReactivatorsKorabecny, Jan ; Soukup, Ondrej ; Dolezal, Rafael ; Spilovska, Katarina ; Nepovimova, Eugenie ; Andrs, Martin ; Nguyen, Thuy Duong ; Jun, Daniel ; Musilek, Kamil ; Kucerova-Chlupacova, Marta ; Kuca, KamilMini reviews in medicinal chemistry, 2014-01, Vol.14 (3), p.215-221 [Periódico revisado por pares]Netherlands: Bentham Science Publishers LtdTexto completo disponível |
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9 |
Material Type: Artigo
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A Review of the Synthesis of Quaternary Acetylcholinesterase ReactivatorsMalinak, David ; Korabecny, Jan ; Soukup, Ondrej ; Gorecki, Lukas ; Nepovimova, Eugenie ; Psotka, Miroslav ; Dolezal, Rafael ; Nguyen, Thuy D. ; Mezeiova, Eva ; Musilek, Kamil ; Kuca, KamilCurrent organic chemistry, 2018-01, Vol.22 (16), p.1619-1648 [Periódico revisado por pares]Bentham Science Publishers LtdTexto completo disponível |
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10 |
Material Type: Artigo
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In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain BarrierChlebek, Jakub ; Korábečný, Jan ; Doležal, Rafael ; Štěpánková, Šárka ; Pérez, Daniel I ; Hošťálková, Anna ; Opletal, Lubomír ; Cahlíková, Lucie ; Macáková, Kateřina ; Kučera, Tomáš ; Hrabinová, Martina ; Jun, DanielMolecules (Basel, Switzerland), 2019-04, Vol.24 (7), p.1340 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |