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1 |
Material Type: Artigo
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Minimum structural requirements for inhibitors of the zinc finger protein TRAF6Radwan, Mohamed O. ; Koga, Ryoko ; Hida, Tomohiro ; Ejima, Tomohiko ; Kanemaru, Yosuke ; Tateishi, Hiroshi ; Okamoto, Yoshinari ; Inoue, Jun-ichiro ; Fujita, Mikako ; Otsuka, MasamiBioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2162-2167 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Structural simplification of evodiamine: Discovery of novel tetrahydro-[beta]-carboline derivatives as potent antitumor agentsSheng, Chunquan ; Zhu, Fugui ; Chen, Shuqiang ; Dong, Guoqiang ; Liu, Dan ; Wan, Kun ; Huang, Yahui ; Ma, ZonglinBioorganic & medicinal chemistry letters, 2021-05, Vol.40 [Periódico revisado por pares]Elsevier B.VTexto completo disponível |
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Material Type: Artigo
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Design, synthesis and bioactivity evaluation of novel pyrazole linked phenylthiazole derivatives in context of antibacterial activityPatel, Bhautikkumar ; Zunk, Matthew ; Grant, Gary ; Rudrawar, SantoshBioorganic & medicinal chemistry letters, 2021-05, Vol.39, p.127853-127853, Article 127853 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Sulfonamide derivatives as multi-target agents for complex diseasesApaydın, Sinem ; Török, MariannaBioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2042-2050 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and biological evaluation of novel 4,7-disubstituted coumarins as selective tumor-associated carbonic anhydrase IX and XII inhibitorsChandra, K. Muni ; Goud, Nerella Sridhar ; Arifuddin, Mohammed ; Alvala, Mallika ; Alvala, Ravi ; Angeli, Andrea ; Supuran, Claudiu T.Bioorganic & medicinal chemistry letters, 2021-05, Vol.39, p.127877-127877, Article 127877 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Pyridones in drug discovery: Recent advancesZhang, Yun ; Pike, AndrewBioorganic & medicinal chemistry letters, 2021-04, Vol.38, p.127849-127849, Article 127849 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Selective degradation of CDK6 by a palbociclib based PROTACRana, Sandeep ; Bendjennat, Mourad ; Kour, Smit ; King, Hannah M. ; Kizhake, Smitha ; Zahid, Muhammad ; Natarajan, AmarnathBioorganic & medicinal chemistry letters, 2019-06, Vol.29 (11), p.1375-1379 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Recent advances in natural antifungal flavonoids and their derivativesJin, Yong-ShengBioorganic & medicinal chemistry letters, 2019-10, Vol.29 (19), p.126589-126589, Article 126589 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
9 |
Material Type: Artigo
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The SARS-CoV-2 main protease as drug targetUllrich, Sven ; Nitsche, ChristophBioorganic & medicinal chemistry letters, 2020-09, Vol.30 (17), p.127377-127377, Article 127377 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
10 |
Material Type: Artigo
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A first-in-class clinical G-quadruplex-targeting drug. The bench-to-bedside translation of the fluoroquinolone QQ58 to CX-5461 (Pidnarulex)Xu, Hong ; Hurley, Laurence H.Bioorganic & medicinal chemistry letters, 2022-12, Vol.77, p.129016-129016, Article 129016 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |