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1
Antibacterial and antibiotic modifying activity, ADMET study and molecular docking of synthetic chalcone (E)-1-(2-hydroxyphenyl)-3-(2,4-dimethoxy-3-methylphenyl)prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps
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Antibacterial and antibiotic modifying activity, ADMET study and molecular docking of synthetic chalcone (E)-1-(2-hydroxyphenyl)-3-(2,4-dimethoxy-3-methylphenyl)prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps

Rocha, Janaína Esmeraldo ; de Freitas, Thiago Sampaio ; da Cunha Xavier, Jayze ; Pereira, Raimundo Luiz Silva ; Junior, Francisco Nascimento Pereira ; Nogueira, Carlos Emídio Sampaio ; Marinho, Márcia Machado ; Bandeira, Paulo Nogueira ; de Oliveira, Mateus Rodrigues ; Marinho, Emmanuel Silva ; Teixeira, Alexandre Magno Rodrigues ; dos Santos, Hélcio Silva ; Coutinho, Henrique Douglas Melo

Biomedicine & pharmacotherapy, 2021-08, Vol.140, p.111768, Article 111768 [Periódico revisado por pares]

Elsevier Masson SAS

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2
Aminophenyl chalcones potentiating antibiotic activity and inhibiting bacterial efflux pump
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Aminophenyl chalcones potentiating antibiotic activity and inhibiting bacterial efflux pump

Siqueira, Marina Micaele Rodrigues ; Freire, Paulo de Tarso Cavalcante ; Cruz, Beatriz Gonçalves ; de Freitas, Thiago Sampaio ; Bandeira, Paulo Nogueira ; Silva dos Santos, Hélcio ; Nogueira, Carlos Emidío Sampaio ; Teixeira, Alexandre Magno Rodrigues ; Pereira, Raimundo Luiz Silva ; Xavier, Jayze da Cunha ; Campina, Fábia Ferreira ; dos Santos Barbosa, Cristina Rodrigues ; Neto, José Bezerra de Araújo ; da Silva, Maria Milene Costa ; Siqueira-Júnior, José Pinto ; Douglas Melo Coutinho, Henrique

European journal of pharmaceutical sciences, 2021-03, Vol.158, p.105695-105695, Article 105695 [Periódico revisado por pares]

Netherlands: Elsevier B.V

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3
Structural characterization, DFT calculations, ADMET studies, antibiotic potentiating activity, evaluation of efflux pump inhibition and molecular docking of chalcone (E)-1-(2-hydroxy-3,4,6-trimethoxyphenyl)-3-(4-methoxyphenyl)prop-2-en-1-one
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Structural characterization, DFT calculations, ADMET studies, antibiotic potentiating activity, evaluation of efflux pump inhibition and molecular docking of chalcone (E)-1-(2-hydroxy-3,4,6-trimethoxyphenyl)-3-(4-methoxyphenyl)prop-2-en-1-one

da Cunha Xavier, Jayze ; Almeida-Neto, Francisco Wagner de Queiroz ; da Silva, Priscila Teixeira ; de Sousa, Amanda Pereira ; Marinho, Emmanuel Silva ; Marinho, Márcia Machado ; Rocha, Janaina Esmeraldo ; Freitas, Priscila Ramos ; de Araújo, Ana Carolina Justino ; Freitas, Thiago Santiago ; Nogueira, Carlos Emídio Sampaio ; de Lima-Neto, Pedro ; Bandeira, Paulo Nogueira ; Teixeira, Alexandre Magno Rodrigues ; Coutinho, Henrique Douglas Melo ; dos Santos, Hélcio Silva

Journal of molecular structure, 2021-03, Vol.1227, p.129692, Article 129692 [Periódico revisado por pares]

Elsevier B.V

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4
Spectroscopic analysis by NMR, FT-Raman, ATR-FTIR, and UV-Vis, evaluation of antimicrobial activity, and in silico studies of chalcones derived from 2-hydroxyacetophenone
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Spectroscopic analysis by NMR, FT-Raman, ATR-FTIR, and UV-Vis, evaluation of antimicrobial activity, and in silico studies of chalcones derived from 2-hydroxyacetophenone

Xavier, Jayze da Cunha ; de Almeida-Neto, Francisco W.Q. ; Rocha, Janaína E. ; Freitas, Thiago S. ; Freitas, Priscila R. ; de Araújo, Ana C.J. ; da Silva, Priscila T. ; Nogueira, Carlos E.S. ; Bandeira, Paulo N. ; Marinho, Márcia M. ; Marinho, Emmanuel S. ; Kumar, Nitin ; Barreto, Antônio C.H. ; Coutinho, Henrique D.M. ; Julião, Murilo S.S. ; dos Santos, Hélcio S. ; Teixeira, Alexandre M.R.

Journal of molecular structure, 2021-10, Vol.1241, p.130647, Article 130647 [Periódico revisado por pares]

Elsevier B.V

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5
Antibacterial and antibiotic modifying activity of chalcone (2E)-1-(4′-aminophenyl)-3-(4-methoxyphenyl)-prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps: In vitro and in silico approaches
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Artigo
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Antibacterial and antibiotic modifying activity of chalcone (2E)-1-(4′-aminophenyl)-3-(4-methoxyphenyl)-prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps: In vitro and in silico approaches

Silva, Jacilene ; Esmeraldo Rocha, Janaína ; da Cunha Xavier, Jayze ; Sampaio de Freitas, Thiago ; Douglas Melo Coutinho, Henrique ; Nogueira Bandeira, Paulo ; Rodrigues de Oliveira, Mateus ; Nunes da Rocha, Matheus ; Machado Marinho, Emanuelle ; de Kassio Vieira Monteiro, Norberto ; Ribeiro, Lyanna Rodrigues ; Róseo Paula Pessoa Bezerra de Menezes, Ramon ; Machado Marinho, Márcia ; Magno Rodrigues Teixeira, Alexandre ; Silva dos Santos, Hélcio ; Silva Marinho, Emmanuel

Microbial pathogenesis, 2022-08, Vol.169, p.105664-105664, Article 105664 [Periódico revisado por pares]

Elsevier Ltd

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6
Spectroscopic characterization and efflux pump modulation of a thiophene curcumin derivative
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Spectroscopic characterization and efflux pump modulation of a thiophene curcumin derivative

Oliveira, Mauro M. ; Santos, Helcio S. ; Coutinho, Henrique D.M. ; Bandeira, Paulo N. ; da Silva, Priscila T. ; Freitas, Thiago S. ; Rocha, Janaina E. ; Xavier, Jayze C. ; Campina, Fabia F. ; Barbosa, Cristina R.S. ; Araújo Neto, José B. ; Pereira, Raimundo L.S. ; Silva, Maria M.C. ; Muniz, Débora F. ; Teixeira, Alexandre M.R. ; Frota, Vanessa M. ; Rodrigues, Tigressa H.S. ; Amado, Ana M. ; Marques, Maria P.M. ; Batista de Carvalho, Luis A.E. ; Nogueira, Carlos E.S.

Journal of molecular structure, 2020-09, Vol.1215, p.128291, Article 128291 [Periódico revisado por pares]

Elsevier B.V

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7
Structural characterization, antibacterial activity and NorA efflux pump inhibition of flavonoid fisetinidol
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Structural characterization, antibacterial activity and NorA efflux pump inhibition of flavonoid fisetinidol

da Silva, Horlando Carlota ; Leal, Antonio Linkoln Alves Borges ; de Oliveira, Mauro Macedo ; Barreto, Humberto Medeiros ; Coutinho, Henrique Douglas Melo ; dos Santos, Hélcio Silva ; Santiago, Gilvandete Maria Pinheiro ; de Freitas, Thiago Sampaio ; Lima, Igor Kleber Campos ; Teixeira, Alexandre Magno Rodrigues ; Nogueira, Carlos Emídio Sampaio

South African journal of botany, 2020-08, Vol.132, p.140-145 [Periódico revisado por pares]

Elsevier B.V

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