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1 |
Material Type: Artigo
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Novel Pieces for the Emerging Picture of Sulfoximines in Drug Discovery: Synthesis and Evaluation of Sulfoximine Analogues of Marketed Drugs and Advanced Clinical CandidatesSirvent, Juan Alberto ; Lücking, UlrichChemMedChem, 2017-04, Vol.12 (7), p.487-501 [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 InhibitorsNuti, Elisa ; Cuffaro, Doretta ; D'Andrea, Felicia ; Rosalia, Lea ; Tepshi, Livia ; Fabbi, Marina ; Carbotti, Grazia ; Ferrini, Silvano ; Santamaria, Salvatore ; Camodeca, Caterina ; Ciccone, Lidia ; Orlandini, Elisabetta ; Nencetti, Susanna ; Stura, Enrico A. ; Dive, Vincent ; Rossello, ArmandoChemMedChem, 2016-08, Vol.11 (15), p.1626-1637 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)Scott, William J. ; Hentemann, Martin F. ; Rowley, R. Bruce ; Bull, Cathy O. ; Jenkins, Susan ; Bullion, Ann M. ; Johnson, Jeffrey ; Redman, Anikó ; Robbins, Arthur H. ; Esler, William ; Fracasso, R. Paul ; Garrison, Timothy ; Hamilton, Mark ; Michels, Martin ; Wood, Jill E. ; Wilkie, Dean P. ; Xiao, Hong ; Levy, Joan ; Stasik, Enrico ; Liu, Ningshu ; Schaefer, Martina ; Brands, Michael ; Lefranc, JulienChemMedChem, 2016-07, Vol.11 (14), p.1517-1530 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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Half-Life Extension of Biopharmaceuticals using Chemical Methods: Alternatives to PEGylationvan Witteloostuijn, Søren B. ; Pedersen, Søren L. ; Jensen, Knud J.ChemMedChem, 2016-11, Vol.11 (22), p.2474-2495 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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Fighting Cancer with Transition Metal Complexes: From Naked DNA to Protein and Chromatin Targeting StrategiesPalermo, Giulia ; Magistrato, Alessandra ; Riedel, Tina ; von Erlach, Thibaud ; Davey, Curt A. ; Dyson, Paul J. ; Rothlisberger, UrsulaChemMedChem, 2016-06, Vol.11 (12), p.1199-1210 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
6 |
Material Type: Artigo
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Antioxidant Activity, Acetylcholinesterase, and Carbonic Anhydrase Inhibitory Properties of Novel Ureas Derived from PhenethylaminesAksu, Kadir ; Özgeriş, Bünyamin ; Taslimi, Parham ; Naderi, Ali ; Gülçin, İlhami ; Göksu, SüleymanArchiv der Pharmazie (Weinheim), 2016-12, Vol.349 (12), p.944-954 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
7 |
Material Type: Artigo
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Efficient Inhibition of Telomerase by Nickel-Salophen ComplexesLecarme, Laureline ; Prado, Enora ; De Rache, Aurore ; Nicolau-Travers, Marie-Laure ; Gellon, Gisèle ; Dejeu, Jérôme ; Lavergne, Thomas ; Jamet, Hélène ; Gomez, Dennis ; Mergny, Jean-Louis ; Defrancq, Eric ; Jarjayes, Olivier ; Thomas, FabriceChemMedChem, 2016-06, Vol.11 (11), p.1133-1136 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
8 |
Material Type: Artigo
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Photodelivery of CO by Designed PhotoCORMs: Correlation between Absorption in the Visible Region and Metal-CO Bond Labilization in Carbonyl ComplexesChakraborty, Indranil ; Carrington, Samantha J. ; Mascharak, Pradip K.ChemMedChem, 2014-06, Vol.9 (6), p.1266-1274 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
9 |
Material Type: Artigo
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Theranostic Nanoparticles Loaded with Imaging Probes and Rubrocurcumin for Combined Cancer Therapy by Folate Receptor TargetingAlberti, Diego ; Protti, Nicoletta ; Franck, Morgane ; Stefania, Rachele ; Bortolussi, Silva ; Altieri, Saverio ; Deagostino, Annamaria ; Aime, Silvio ; Geninatti Crich, SimonettaChemMedChem, 2017-04, Vol.12 (7), p.502-509 [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
10 |
Material Type: Artigo
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Anticancer Therapeutics That Target Selenoenzymes: Synthesis, Characterization, in vitro Cytotoxicity, and Thioredoxin Reductase Inhibition of a Series of Gold(I) Complexes Containing Hydrophilic Phosphine LigandsVergara, Elena ; Casini, Angela ; Sorrentino, Francesca ; Zava, Olivier ; Cerrada, Elena ; Rigobello, Maria Pia ; Bindoli, Alberto ; Laguna, Mariano ; Dyson, Paul J.ChemMedChem, 2010-01, Vol.5 (1), p.96-102 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |