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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxam i des as potent and selective CB sub(2) receptor agonists

Han, Sangdon ; Thoresen, Lars ; Zhu, Xiuwen ; Narayanan, Sanju ; Jung, Jae-Kyu ; Strah-Pleynet, Sonja ; Decaire, Marc ; Choi, Karoline ; Xiong, Yifeng ; Yue, Dawei ; Semple, Graeme ; Thatte, Jayant ; Solomon, Michelle ; Fu, Lixia ; Whelan, Kevin ; Al-Shamma, Hussien ; Gatlin, Joel ; Chen, Ruoping ; Dang, Huong ; Pride, Cameron ; Gaidarov, Ibragim ; Unett, David J ; Behan, Dominic P ; Sadeque, Abu ; Usmani, Khawja A ; Chen, Chuan ; Edwards, Jeffrey ; Morgan, Michael ; Jones, Robert M

Bioorganic & medicinal chemistry letters, 2015-01, Vol.25 (2), p.322-326 [Periódico revisado por pares]

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