Synthesis and Biological Evaluation of the 1‑Arylpyrazole Class of σ1 Receptor Antagonists: Identification of 4‑{2-[5-Methyl-1-(naphthalen-2-yl)‑1H‑pyrazol-3-yloxy]ethyl}morpholine (S1RA, E‑52862)

Díaz, José Luis ; Cuberes, Rosa ; Berrocal, Joana ; Contijoch, Montserrat ; Christmann, Ute ; Fernández, Ariadna ; Port, Adriana ; Holenz, Jörg ; Buschmann, Helmut ; Laggner, Christian ; Serafini, Maria Teresa ; Burgueño, Javier ; Zamanillo, Daniel ; Merlos, Manuel ; Vela, José Miguel ; Almansa, Carmen

Journal of medicinal chemistry, 2012-10, Vol.55 (19), p.8211-8224 [Periódico revisado por pares]

American Chemical Society

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