Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)
Scott, William J. ; Hentemann, Martin F. ; Rowley, R. Bruce ; Bull, Cathy O. ; Jenkins, Susan ; Bullion, Ann M. ; Johnson, Jeffrey ; Redman, Anikó ; Robbins, Arthur H. ; Esler, William ; Fracasso, R. Paul ; Garrison, Timothy ; Hamilton, Mark ; Michels, Martin ; Wood, Jill E. ; Wilkie, Dean P. ; Xiao, Hong ; Levy, Joan ; Stasik, Enrico ; Liu, Ningshu ; Schaefer, Martina ; Brands, Michael ; Lefranc, Julien
ChemMedChem, 2016-07, Vol.11 (14), p.1517-1530 [Periódico revisado por pares]Germany: Blackwell Publishing Ltd
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